SCHEMBL24521577

SCHEMBL24521577

CC(C)(C)OC(=O)Oc1ccc(CCC(=O)NCc2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC10 Q969S8 1/20 0.49
HDAC11 Q96DB2 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
ALDH1A1 P00352 3/20 0.46
TP53 P04637 3/20 0.46
MAPK14 Q16539 1/20 0.45
FFAR1 O14842 1/20 0.44
PPARA Q07869 1/20 0.43
ELANE P08246 1/20 0.43
GAA P10253 1/20 0.42
LTA4H P09960 1/20 0.42
EPHX2 P34913 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24521562 0.88 FFAR1 (0.49) MAPK14FFAR1
SCHEMBL24521601 0.83 GAA (0.54) HDAC1HDAC8MEN1KMT2AALDH1A1
SCHEMBL24521503 0.78 MTOR (0.62) HDAC3HDAC1HDAC2HDAC10HDAC11
SCHEMBL30791534 0.78 TRPV1 (0.63) HDAC3HDAC1HDAC2HDAC10HDAC11
SCHEMBL22547959 0.77 HDAC3 (0.61) HDAC3HDAC1HDAC2HDAC10HDAC11
SCHEMBL29052292 0.77 CTSS (0.53) HDAC8PPARA
SCHEMBL24521579 0.77 CTSS (0.53) HDAC8PPARA
SCHEMBL4574985 0.75 LSS (0.52) HDAC3HDAC1HDAC2HDAC10HDAC11
SCHEMBL29059895 0.75 ELANE (0.57) KMT2AALDH1A1FFAR1PPARAELANE
SCHEMBL29562370 0.75 ELANE (0.57) FFAR1ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4015501-A1 N-BENZYL-ALPHA-AMINOAMIDES AS ANAPHASE-PROMOTING COMPLEX/CYCLOSOME (APC/C) INHIBITORS Consejo Superior de Investigaciones Científicas (CSIC) (ES) 2022-06-22 EP disclosed