SCHEMBL24521880

SCHEMBL24521880

COc1ccc(C(CC(=O)OC(C)(C)C)N/C=C\C(=N)CCCc2ccc3cccnc3n2)cn1

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SUCNR1 Q9BXA5 14/20 0.38
OXGR1 Q96P68 2/20 0.38
ITGB3 P05106 6/20 0.37
ITGAV P06756 6/20 0.37
BDKRB1 P46663 1/20 0.34
ITGB6 P18564 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20153460 0.91 SUCNR1 (0.39) SUCNR1OXGR1ITGB3ITGAVBDKRB1
SCHEMBL20153379 0.88 ITGB3 (0.33) SUCNR1OXGR1ITGB3ITGAVITGB6
SCHEMBL20153358 0.86 ITGB3 (0.33) ITGB3ITGAV
SCHEMBL24521878 0.84 ITGAV (0.57) ITGB3ITGAVITGB6
SCHEMBL24521828 0.82 ITGAV (0.60) ITGB3ITGAVITGB6
SCHEMBL21311584 0.78 ITGB3 (0.38) SUCNR1OXGR1ITGB3ITGAVBDKRB1
SCHEMBL20153461 0.77 ITGAV (0.59) ITGB3ITGAVITGB6
SCHEMBL20153349 0.74 ITGAV (0.64) ITGB3ITGAVITGB6
SCHEMBL20153385 0.74 ITGAV (0.64) ITGB3ITGAVITGB6
SCHEMBL24521903 0.74 ITGAV (0.61) ITGB3ITGAVITGB6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538525-B1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2022-06-22 EP disclosed