SCHEMBL20153358

SCHEMBL20153358

COc1ccc(C(CC(=O)OC(C)(C)C)N/C=C\C(=N)CCCC(C)=O)cn1

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 11/20 0.33
ITGAV P06756 10/20 0.33
KCNK3 O14649 5/20 0.33
KCNK9 Q9NPC2 1/20 0.33
ITGA2B P08514 1/20 0.31
NR3C1 P04150 1/20 0.30
ITGB1 P05556 1/20 0.30
ITGA4 P13612 1/20 0.30
NNMT P40261 1/20 0.30
TRPM8 Q7Z2W7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24521880 0.86 SUCNR1 (0.38) ITGB3ITGAV
SCHEMBL24521878 0.81 ITGAV (0.57) ITGB3ITGAVITGA2BITGB1
SCHEMBL24521828 0.81 ITGAV (0.60) ITGB3ITGAVITGA2BITGB1
SCHEMBL20153459 0.78 KCNK3 (0.34) ITGB3ITGAVKCNK3KCNK9ITGA2B
SCHEMBL20153460 0.76 SUCNR1 (0.39) ITGB3ITGAV
SCHEMBL20153379 0.76 ITGB3 (0.33) ITGB3ITGAVKCNK3TRPM8
SCHEMBL17262997 0.72 ADRB3 (0.38) ITGB3ITGAVKCNK3KCNK9NR3C1
SCHEMBL13719466 0.72 ADRB3 (0.38) ITGB3ITGAVKCNK3KCNK9NR3C1
SCHEMBL20153461 0.72 ITGAV (0.59) ITGB3ITGAVITGA2BITGB1
SCHEMBL20087016 0.72 ADRB3 (0.38) ITGB3ITGAVKCNK3KCNK9NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538525-B1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2022-06-22 EP disclosed
WO-2018089353-A1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed