SCHEMBL24521912

SCHEMBL24521912

COc1ccc(C(CC(=O)O)/C(C=N)=C/NCCCCc2ccc3c(n2)NCCC3)cc1F

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 20/20 0.59
ITGAV P06756 20/20 0.59
ITGB6 P18564 11/20 0.59
ITGA2B P08514 2/20 0.59
ITGB5 P18084 11/20 0.56
ITGB8 P26012 9/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20153331 0.86 ITGAV (0.65) ITGB3ITGAVITGB6ITGA2BITGB5
SCHEMBL20153363 0.84 ITGAV (0.64) ITGB3ITGAVITGB6ITGA2BITGB5
SCHEMBL24521899 0.81 ITGB3 (0.67) ITGB3ITGAVITGB6ITGA2BITGB5
SCHEMBL23912903 0.80 ITGB3 (0.54) ITGB3ITGAVITGB6ITGA2BITGB5
SCHEMBL20156291 0.80 ITGB3 (0.62) ITGB3ITGAVITGB6ITGA2BITGB5
SCHEMBL21294628 0.80 ITGB3 (0.71) ITGB3ITGAVITGB6ITGA2BITGB5
SCHEMBL24521917 0.79 ITGB3 (0.62) ITGB3ITGAVITGB6ITGA2BITGB5
SCHEMBL23912864 0.78 ITGB3 (0.60) ITGB3ITGAVITGB6ITGA2BITGB5
SCHEMBL21294658 0.78 ITGAV (0.67) ITGB3ITGAVITGB6ITGA2BITGB5
SCHEMBL21294650 0.78 ITGAV (0.67) ITGB3ITGAVITGB6ITGA2BITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538525-B1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2022-06-22 EP disclosed