SCHEMBL24528591

SCHEMBL24528591

CN(C)CCC/N=C\c1ccc(-c2nc(NCCCN(C)C)nc3ccsc23)cc1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.41
ADORA2A P29274 6/20 0.41
ADORA1 P30542 6/20 0.41
RAD52 P43351 2/20 0.37
TRIM58 Q8NG06 2/20 0.36
KCNH2 Q12809 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24528628 0.85 ADORA2A (0.34) ADORA2AADORA1RAD52
SCHEMBL24528642 0.84 SCN9A (0.41) SCN9ATRIM58
SCHEMBL24528590 0.84 ADORA2A (0.40) ADORA2AADORA1
SCHEMBL24528664 0.70 ADORA2A (0.34) ADORA2A
SCHEMBL24528643 0.69 NUDT1 (0.38)
SCHEMBL24528587 0.68 KDM4E (0.40) RAD52
SCHEMBL29681009 0.68 KDM4E (0.40) RAD52
SCHEMBL3681700 0.65 ADORA2A (0.73) SCN9AADORA2AADORA1RAD52
SCHEMBL24528588 0.64 ALDH1A1 (0.36)
SCHEMBL24528635 0.63 BPTF (0.38) ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed