SCHEMBL24528640

SCHEMBL24528640

CN(C)CCCC/N=C\c1ccc(-c2nc(-c3ccc(/C=N/CCCCN(C)C)cc3)nc3c2N(C)CN3c2ccccc2)cc1

nearest known ligand 0.32

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 2/20 0.32
MAOB P27338 1/20 0.31
THRB P10828 1/20 0.31
NPY1R P25929 1/20 0.31
NPY2R P49146 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
MEN1 O00255 1/20 0.30
PSMD14 O00487 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24528693 0.99 TLR9 (0.31) TLR9MAOBTHRBNPY1RNPY2R
SCHEMBL24528701 0.88 KDM4E (0.33) MAOBALDH1A1LMNAMEN1PSMD14
SCHEMBL24528686 0.86 RAB9A (0.35) TLR9L3MBTL1ALDH1A1
SCHEMBL24528611 0.77 ADK (0.35) L3MBTL1ALDH1A1LMNAMEN1KMT2A
SCHEMBL24528695 0.75 KDM4E (0.34) TLR9MAOBTHRBNPY1RNPY2R
SCHEMBL24528639 0.75 ATM (0.37) TLR9MAOBALDH1A1LMNA
SCHEMBL29680708 0.75 GSK3B (0.41) ALDH1A1MEN1KMT2A
SCHEMBL24528677 0.75 KDM4E (0.34) TLR9MAOBALDH1A1LMNA
SCHEMBL29680812 0.74 GSK3B (0.40) ALDH1A1MEN1KMT2A
SCHEMBL24528655 0.73 KDM4E (0.34) TLR9THRBNPY1RNPY2RL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed