SCHEMBL24528686

SCHEMBL24528686

CN1CCN(CCCC/N=C\c2ccc(-c3nc(-c4ccc(/C=N/CCCCN5CCN(C)CC5)cc4)nc4c3N(C)CN4c3ccccc3)cc2)CC1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.35
POLB P06746 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.33
NPC1 O15118 2/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
AVPR1A P37288 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
TLR9 Q9NR96 5/20 0.33
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24528640 0.86 TLR9 (0.32) ALDH1A1L3MBTL1TLR9
SCHEMBL24528693 0.85 TLR9 (0.31) ALDH1A1L3MBTL1TLR9
SCHEMBL24528690 0.78 TLR9 (0.41) RAB9ASMN1; SMN2KDM4EALDH1A1NPC1
SCHEMBL24528661 0.78 RAD52 (0.36) RAB9APOLBNPSR1HTTSMN1; SMN2
SCHEMBL29680767 0.78 KDM5B (0.42) KDM4EALDH1A1MAPTMAPK1
SCHEMBL24528701 0.76 KDM4E (0.33) KDM4EALDH1A1
SCHEMBL24528611 0.76 ADK (0.35) RAB9APOLBNPSR1HTTSMN1; SMN2
SCHEMBL24528648 0.76 RAD52 (0.37) RAB9APOLBNPSR1HTTSMN1; SMN2
SCHEMBL29680554 0.76 RAD52 (0.37) RAB9APOLBNPSR1HTTSMN1; SMN2
SCHEMBL24528607 0.73 TLR9 (0.36) RAB9APOLBNPSR1HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed