SCHEMBL24528690

SCHEMBL24528690

CN1CCN(CCCC/N=C\c2ccc(-c3nc(-c4ccc(/C=N/CCCCN5CCN(C)CC5)cc4)nc4c3ncn4-c3ccccc3)cc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 3/20 0.41
AVPR1A P37288 8/20 0.35
AVPR2 P30518 7/20 0.35
RAD52 P43351 1/20 0.35
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
MAPT P10636 1/20 0.34
MAPK1 P28482 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24528661 0.86 RAD52 (0.36) TLR9AVPR1ARAD52NPC1RAB9A
SCHEMBL24528639 0.84 ATM (0.37) TLR9KDM4EALDH1A1
SCHEMBL29680554 0.83 RAD52 (0.37) TLR9AVPR1ARAD52NPC1RAB9A
SCHEMBL24528648 0.83 RAD52 (0.37) TLR9AVPR1ARAD52NPC1RAB9A
SCHEMBL29680767 0.82 KDM5B (0.42) RAD52MAPTMAPK1KDM4EALDH1A1
SCHEMBL24528649 0.79 RAD52 (0.34) TLR9AVPR1ARAD52NPC1RAB9A
SCHEMBL24528686 0.78 RAB9A (0.35) TLR9AVPR1ANPC1RAB9AMAPT
SCHEMBL24528685 0.75 KDM4E (0.40) TLR9RAD52NPC1RAB9AMAPT
SCHEMBL29681200 0.75 KDM4E (0.40) TLR9RAD52NPC1RAB9AMAPT
SCHEMBL24528659 0.74 ALDH1A1 (0.36) RAD52NPC1RAB9AMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed