SCHEMBL24548618

SCHEMBL24548618

CC(C)c1cc(Oc2c(Cl)cccc2Cl)nnc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 13/20 0.36
THRA P10827 12/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CYP2C9 P11712 1/20 0.33
UGT1A1 P22309 1/20 0.33
ABCG2 Q9UNQ0 1/20 0.33
SLCO1B1 Q9Y6L6 1/20 0.33
ADRA2A P08913 2/20 0.33
ADRA2B P18089 2/20 0.33
ADRA2C P18825 2/20 0.33
HTR1A P08908 1/20 0.33
SLC6A4 P31645 1/20 0.33
ADRA1A P35348 1/20 0.33
OPRK1 P41145 1/20 0.33
KCNH2 Q12809 1/20 0.33
RORC P51449 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2045628 0.85 LMNA (0.33) THRBTHRAKDM4ELMNACYP1A2
SCHEMBL21749438 0.83 THRA (0.38) THRBTHRACYP2C9UGT1A1ABCG2
SCHEMBL29417446 0.83 THRA (0.38) THRBTHRACYP2C9UGT1A1ABCG2
SCHEMBL28564386 0.83 THRA (0.36) THRBTHRACYP2C9UGT1A1ABCG2
SCHEMBL30820597 0.83 THRB (0.39) THRBTHRACYP2C9UGT1A1ABCG2
SCHEMBL13116309 0.83 THRB (0.39) THRBTHRACYP2C9UGT1A1ABCG2
SCHEMBL30398362 0.83 THRA (0.41) THRBTHRACYP2C9UGT1A1ABCG2
SCHEMBL22660386 0.83 THRA (0.41) THRBTHRACYP2C9UGT1A1ABCG2
SCHEMBL21840329 0.83 THRA (0.38) THRBTHRACYP2C9UGT1A1ABCG2
SCHEMBL2049678 0.80 RORC (0.38) THRBKDM4ELMNACYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022127779-A1 SUBSTITUTED PYRIDAZINONE COMPOUND AND USE THEREOF 山东第一医科大学(山东省医学科学院) 2022-06-23 WO disclosed