SCHEMBL2456934

SCHEMBL2456934

CC(O)(c1cc(F)cc(Cl)c1)C(Cl)Cl

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
RAPGEF4 Q8WZA2 3/20 0.33
RAPGEF3 O95398 2/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2449028 0.88 SLC6A3 (0.34)
SCHEMBL9967852 0.76 GABRA1 (0.37) RAPGEF4RAPGEF3
SCHEMBL9152278 0.72 PDE2A (0.38) RAPGEF4RAPGEF3
SCHEMBL2460935 0.72 MEN1 (0.38) MEN1KMT2A
Hydrochloric Acid SCHEMBL31410065 0.71 PDE2A (0.36) RAPGEF4
SCHEMBL1331197 0.69 CHRM3 (0.30)
SCHEMBL7934061 0.69 RAPGEF4 (0.42) RAPGEF4
SCHEMBL9152935 0.66 SLC6A3 (0.41) RAPGEF4RAPGEF3
SCHEMBL1155869 0.64
SCHEMBL1360451 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2367786-A1 NOVEL 1 -ALKYL- 3 -HYDROXY- 3 -PHENYLAZETIDINE DERIVATIVES USEFUL AS MODULATORS OF CORTICAL CATECHOLAMINERGIC NEUROTRANSMISSION NSAB, Filial af NeuroSearch Sweden AB, Sverige (DK) 2011-09-28 EP disclosed
WO-2010058020-A1 NOVEL 1 -ALKYL- 3 -HYDROXY- 3 -PHENYLAZETIDINE DERIVATIVES USEFUL AS MODULATORS OF CORTICAL CATECHOLAMINERGIC NEUROTRANSMISSION NSAB, FILIAL AF NEUROSEARCH SWEDEN AB, SVERIGE (DK) 2010-05-27 WO disclosed