SCHEMBL2460935

SCHEMBL2460935

CC(O)(c1ccc(F)c(F)c1)C(Cl)Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
KCNN4 O15554 1/20 0.38
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
CHRM3 P20309 1/20 0.36
PDE2A O00408 3/20 0.36
CHRNA1 P02708 1/20 0.36
CHRNG P07510 1/20 0.36
CHRNB1 P11230 1/20 0.36
CHRNB2 P17787 1/20 0.36
SLC6A2 P23975 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
SLC6A3 Q01959 1/20 0.36
CHRND Q07001 1/20 0.36
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28091068 0.78 MEN1 (0.41) MEN1KMT2AKCNN4AKR1C3AKR1C2
SCHEMBL27902048 0.77 KCNN4 (0.43) MEN1KMT2AKCNN4AKR1C3AKR1C2
SCHEMBL6967423 0.77 KCNN4 (0.43) MEN1KMT2AKCNN4AKR1C3AKR1C2
SCHEMBL2449028 0.74 SLC6A3 (0.34) CHRM3SLC6A3CES2CES1
SCHEMBL828570 0.72 ALDH1A1 (0.46) MEN1KMT2AKCNN4AKR1C3AKR1C2
SCHEMBL3950869 0.72 ESR1 (0.44) KCNN4AKR1C3AKR1C2CHRM3PDE2A
SCHEMBL2456934 0.72 RAPGEF4 (0.33) MEN1KMT2A
SCHEMBL12238633 0.70 PDE2A (0.41) MEN1KMT2AAKR1C3AKR1C2PDE2A
SCHEMBL7225768 0.70 KCNN4 (0.42) MEN1KMT2AKCNN4AKR1C3AKR1C2
SCHEMBL21229776 0.69 KCNN4 (0.45) MEN1KMT2AKCNN4AKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2367786-A1 NOVEL 1 -ALKYL- 3 -HYDROXY- 3 -PHENYLAZETIDINE DERIVATIVES USEFUL AS MODULATORS OF CORTICAL CATECHOLAMINERGIC NEUROTRANSMISSION NSAB, Filial af NeuroSearch Sweden AB, Sverige (DK) 2011-09-28 EP disclosed
WO-2010058020-A1 NOVEL 1 -ALKYL- 3 -HYDROXY- 3 -PHENYLAZETIDINE DERIVATIVES USEFUL AS MODULATORS OF CORTICAL CATECHOLAMINERGIC NEUROTRANSMISSION NSAB, FILIAL AF NEUROSEARCH SWEDEN AB, SVERIGE (DK) 2010-05-27 WO disclosed