SCHEMBL24573233

SCHEMBL24573233

COc1cc2c(Br)c[nH]c2c(F)c1Cl

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
ALOX5 P09917 1/20 0.32
PTGS2 P35354 1/20 0.32
SRC P12931 1/20 0.31
GSK3B P49841 1/20 0.31
EGFR P00533 1/20 0.31
MTNR1A P48039 2/20 0.31
MTNR1B P49286 2/20 0.31
HTR1A P08908 1/20 0.31
IDO1 P14902 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
KMT2A Q03164 1/20 0.30
POLB P06746 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29735061 0.74 ROCK2 (0.40)
SCHEMBL10905707 0.69 MTNR1A (0.65) MTNR1AMTNR1BHTR1AMEN1ALDH1A1
SCHEMBL29361577 0.69 AR (0.42)
SCHEMBL7054082 0.69 MTNR1A (0.66) MTNR1AMTNR1BMEN1KMT2A
SCHEMBL24572813 0.68 MAPT (0.48) ALOX5PTGS2MAPTPOLBL3MBTL1
SCHEMBL24572812 0.68 TNF (0.43) MEN1KMT2APOLB
SCHEMBL27509094 0.67 MTNR1A (0.44) PDE3BPDE3AGSK3BEGFRMTNR1A
SCHEMBL3309764 0.66 CA2 (0.45) MTNR1AMTNR1BALDH1A1MAPT
SCHEMBL13729900 0.66 GSK3B (0.40) PDE3BPDE3AGSK3BMTNR1AMTNR1B
SCHEMBL2883982 0.65 NQO2 (0.38) ALOX5PTGS2MEN1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12404261-B2 Compounds and compositions for treating conditions associated with cGAS NOVARTIS AG (CH) 2025-09-02 US disclosed
CN-116635382-A Indole derivatives useful for treating cGAS-related disorders 诺华股份有限公司 2023-08-22 CN disclosed
US-20230085472-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH cGAS NOVARTIS PHARMA AG (CH) 2023-03-16 US disclosed
WO-2022137085-A1 INDOLE DERIVATIVES USEFUL IN TREATING CONDITIONS ASSOCIATED WITH CGAS NOVARTIS AG (CH) 2022-06-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12404261-B2 Compounds and compositions for treating conditions associated with cGAS CGAS, TDP1, IAPP PDE3B 129/4885PDE3A 91/4885ALOX5 2978/4885
US-20230085472-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH cGAS CGAS, TDP1, IAPP PDE3B 129/4885PDE3A 91/4885ALOX5 2978/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.