SCHEMBL2460997

SCHEMBL2460997

Brc1cccc(C2(Cc3ccccc3)C=NC=N2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.41
MAOB P27338 2/20 0.36
APP P05067 2/20 0.33
TAAR1 Q96RJ0 3/20 0.33
IDO1 P14902 2/20 0.32
AGXT P21549 2/20 0.32
KDM1A O60341 3/20 0.32
RCOR1 Q9UKL0 2/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GABRG2 P18507 2/20 0.31
GABRB3 P28472 2/20 0.31
GABRA5 P31644 2/20 0.31
GABRA3 P34903 2/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27708670 0.69 CHRNA1 (0.35) MEN1KMT2AGABRG2GABRB3GABRA5
SCHEMBL27286322 0.66 ALDH1A1 (0.33)
SCHEMBL27589212 0.66 MAOA (0.38) MAOBIDO1KDM1A
SCHEMBL28746800 0.65 ALDH1A1 (0.32)
SCHEMBL946696 0.64 BACE1 (0.46) NPSR1MAOBAPPTAAR1IDO1
SCHEMBL4717 0.59 CALM1 (0.57) MAOBTAAR1IDO1AGXTKDM1A
SCHEMBL9660784 0.59 TAAR1 (0.65) MAOBTAAR1IDO1AGXTKDM1A
SCHEMBL31499406 0.59 CALM1 (0.57) MAOBTAAR1IDO1AGXTKDM1A
SCHEMBL4795297 0.58 MAOA (0.40) MAOBIDO1AGXTKDM1A
SCHEMBL28239960 0.58 ALDH1A1 (0.44) TAAR1IDO1AGXT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2365748-A1 IMIDAZOISOINDOLE NEUROPEPTIDE S RECEPTOR ANTAGONISTS Merck Sharp & Dohme Corp. (US) 2011-09-21 EP claimed
WO-2010056567-A1 IMIDAZOISOINDOLE NEUROPEPTIDE S RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2010-05-20 WO claimed