SCHEMBL24628458

SCHEMBL24628458

Cc1cc(Br)cc(COc2cccc(NC(=O)c3ccc(-c4ccc(O)cc4)cc3)c2)c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 7/20 0.53
ALDH1A1 P00352 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
NPC1 O15118 3/20 0.52
RAB9A P51151 3/20 0.52
TRPV1 Q8NER1 1/20 0.51
TP53 P04637 3/20 0.49
MAPT P10636 2/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
MAOB P27338 1/20 0.48
RXFP1 Q9HBX9 1/20 0.48
MAPK1 P28482 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26828942 0.83 MCHR1 (0.50) NR1H4ALDH1A1NPC1RAB9AMAPT
SCHEMBL26897513 0.82 NR1H4 (0.48) NR1H4ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL24628454 0.82 MCHR1 (0.50) NR1H4MAPT
SCHEMBL24628824 0.81 SIRT2 (0.53) NR1H4ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL26829283 0.77 MAPT (0.49) NR1H4ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL24628602 0.75 MEN1 (0.67) ALDH1A1NPC1RAB9ATP53MAPT
SCHEMBL26815658 0.75 RAB9A (0.66) ALDH1A1NPC1RAB9ATP53MAPT
SCHEMBL21768134 0.75 THRB (0.61) NR1H4ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL11550139 0.73 NR1H4 (0.81) NR1H4NPC1RAB9AMAPTMEN1
SCHEMBL595158 0.71 MAOB (0.64) NR1H4ALDH1A1NPC1RAB9AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4276092-A1 COMPOUND LIBRARY CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2023-11-15 EP disclosed
WO-2022149617-A1 COMPOUND LIBRARY 中外製薬株式会社 2022-07-14 WO disclosed