SCHEMBL2464513

SCHEMBL2464513

CC(=O)OCc1cc(OC(C)=O)ccn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.48
MAPT P10636 2/20 0.48
CYP3A4 P08684 3/20 0.45
LMNA P02545 4/20 0.41
ALDH1A1 P00352 3/20 0.40
ACHE P22303 2/20 0.38
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
NOS2 P35228 1/20 0.38
GLA P06280 2/20 0.37
F2 P00734 1/20 0.37
HPGD P15428 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ABCB11 O95342 1/20 0.36
ESR1 P03372 1/20 0.36
ADRA2A P08913 1/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
PDE4A P27815 1/20 0.36
ADRA1A P35348 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9814691 0.87 NOS1 (0.53) KDM4EMAPTCYP3A4LMNAALDH1A1
SCHEMBL1982867 0.83 KDM4E (0.47) KDM4EMAPTCYP3A4LMNAALDH1A1
SCHEMBL9566886 0.82 MEN1 (0.41) KDM4EMAPTCYP3A4LMNAALDH1A1
SCHEMBL11369806 0.82 GCK (0.49) KDM4ELMNAALDH1A1SMN1; SMN2NPC1
SCHEMBL17019021 0.81 ALDH1A1 (0.43) KDM4EMAPTCYP3A4LMNAALDH1A1
SCHEMBL509101 0.80 ALDH1A1 (0.42) KDM4ECYP3A4ALDH1A1NOS3NOS1
SCHEMBL9129980 0.80 LNPEP (0.44) CYP2C9LNPEP
SCHEMBL9566840 0.79 KDM4E (0.34) KDM4EMAPTALDH1A1LNPEP
SCHEMBL1477890 0.79 ALDH1A1 (0.43) KDM4EMAPTCYP3A4LMNAALDH1A1
SCHEMBL14086531 0.79 ALDH1A1 (0.41) KDM4EMAPTCYP3A4LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1875239-B1 A METHOD FOR THE PREPARATION OF IMAGING PROBES USING CLICK CHEMISTRY SIEMENS MEDICAL SOLUTIONS (US) 2011-10-05 EP disclosed
EP-1875239-A2 A METHOD FOR THE PREPARATION OF IMAGING PROBES USING CLICK CHEMISTRY Siemens Medical Solutions USA, Inc. (US) 2008-01-09 EP disclosed
US-20060269942-A1 In situ click chemistry method for screening high affinity molecular imaging probes SIEMENS MEDICAL SOLUTIONS USA, INC. 2006-11-30 US disclosed
WO-2006116736-A2 A METHOD FOR THE PREPARATION OF IMAGING PROBES USING CLICK CHEMISTRY SIEMENS MEDICAL SOLUTIONS USA, INC. (US) 2006-11-02 WO disclosed