SCHEMBL24667

SCHEMBL24667

C=C(CCNC(=O)c1ccc2c(c1)/C(=C/c1ccc[nH]1)C(=O)N2)NO

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAK4 O96013 10/20 0.75
CDK1 P06493 1/20 0.63
CCNB1 P14635 1/20 0.63
NEK2 P51955 1/20 0.63
TLK2 Q86UE8 5/20 0.61
PDPK1 O15530 3/20 0.61
JAK3 P52333 2/20 0.61
HDAC3 O15379 1/20 0.56
PDGFRB P09619 1/20 0.56
FLT1 P17948 1/20 0.56
KDR P35968 1/20 0.56
HDAC4 P56524 1/20 0.56
HDAC1 Q13547 1/20 0.56
HDAC7 Q8WUI4 1/20 0.56
HDAC2 Q92769 1/20 0.56
HDAC10 Q969S8 1/20 0.56
HDAC11 Q96DB2 1/20 0.56
HDAC8 Q9BY41 1/20 0.56
HDAC6 Q9UBN7 1/20 0.56
HDAC9 Q9UKV0 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12473990 0.90 PAK4 (0.78) PAK4CDK1CCNB1NEK2TLK2
SCHEMBL12473995 0.90 PAK4 (0.78) PAK4CDK1CCNB1NEK2TLK2
SCHEMBL25738 0.86 PAK4 (0.77) PAK4CDK1CCNB1NEK2TLK2
SCHEMBL5368518 0.81 PAK4 (0.75) PAK4CDK1CCNB1NEK2TLK2
SCHEMBL20937 0.78 PAK4 (0.71) PAK4CDK1CCNB1NEK2TLK2
SCHEMBL12200908 0.78 NEK2 (1.00) PAK4CDK1CCNB1NEK2TLK2
SCHEMBL31061298 0.78 NEK2 (1.00) PAK4CDK1CCNB1NEK2TLK2
SCHEMBL20945 0.77 TLK2 (1.00) PAK4CDK1CCNB1NEK2TLK2
SCHEMBL20944 0.77 TLK2 (1.00) PAK4CDK1CCNB1NEK2TLK2
SCHEMBL5363197 0.77 TLK2 (0.80) PAK4CDK1CCNB1NEK2TLK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012025726-A1 Novel Hybrid Compounds UNIVERSITY OF GREENWICH (GB) 2012-03-01 WO disclosed