SCHEMBL25738

SCHEMBL25738

COC(=O)CCNC(=O)c1ccc2c(c1)/C(=C/c1ccc[nH]1)C(=O)N2

nearest known ligand 0.77

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PAK4 O96013 9/20 0.77
PDPK1 O15530 4/20 0.70
TLK2 Q86UE8 6/20 0.64
CDK1 P06493 1/20 0.64
CCNB1 P14635 1/20 0.64
NEK2 P51955 1/20 0.64
JAK3 P52333 3/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12473995 0.87 PAK4 (0.78) PAK4PDPK1TLK2CDK1CCNB1
SCHEMBL12473990 0.87 PAK4 (0.78) PAK4PDPK1TLK2CDK1CCNB1
SCHEMBL24667 0.86 PAK4 (0.75) PAK4PDPK1TLK2CDK1CCNB1
SCHEMBL5728671 0.82 PDPK1 (1.00) PAK4PDPK1TLK2CDK1CCNB1
SCHEMBL5361523 0.82 PDPK1 (1.00) PAK4PDPK1TLK2CDK1CCNB1
SCHEMBL5368518 0.81 PAK4 (0.75) PAK4PDPK1TLK2CDK1CCNB1
SCHEMBL20937 0.81 PAK4 (0.71) PAK4PDPK1TLK2CDK1CCNB1
SCHEMBL13080513 0.79 TLK2 (1.00) PAK4PDPK1TLK2CDK1CCNB1
SCHEMBL12200908 0.78 NEK2 (1.00) PAK4PDPK1TLK2CDK1CCNB1
SCHEMBL31061298 0.78 NEK2 (1.00) PAK4PDPK1TLK2CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012025726-A1 Novel Hybrid Compounds UNIVERSITY OF GREENWICH (GB) 2012-03-01 WO disclosed