SCHEMBL24669482

SCHEMBL24669482

CC(C)N1CNc2ccncc21

nearest known ligand 0.32

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.32
HTT P42858 1/20 0.32
NCOA1 Q15788 1/20 0.32
NCOA3 Q9Y6Q9 1/20 0.32
NFATC1 O95644 1/20 0.31
GSK3B P49841 1/20 0.31
DYRK1A Q13627 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
TSHR P16473 1/20 0.31
GPBAR1 Q8TDU6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25094288 0.84 HTR2A (0.33) USP2HTTNCOA1NCOA3NFATC1
SCHEMBL7975285 0.83 PDE9A (0.32)
SCHEMBL7977462 0.76 GAA (0.35) GSK3BCYP3A4
SCHEMBL10094143 0.76 BRPF1 (0.42) CYP3A4CYP2D6TSHR
SCHEMBL17953966 0.71 HTR2A (0.40) CYP3A4CYP2D6TSHR
SCHEMBL7033880 0.70 MAPT (0.33) GSK3B
SCHEMBL21234852 0.70 CYP1A2 (0.33) CYP3A4CYP2D6TSHR
SCHEMBL22736596 0.69 SIGMAR1 (0.44) HTTCYP3A4CYP2D6TSHR
SCHEMBL8556566 0.68 GRIA2 (0.35) CYP3A4CYP2D6TSHR
SCHEMBL24597109 0.68 SLC22A12 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022187693-A1 COVALENT CDK2-BINDING COMPOUNDS FOR THERAPEUTIC PURPOSES UMBRA THERAPEUTICS INC. (US) 2022-09-09 WO disclosed