SCHEMBL7977462

SCHEMBL7977462

CN1CNc2ccncc21

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.35
HDAC1 Q13547 1/20 0.34
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
ADORA3 P0DMS8 1/20 0.32
ADORA2A P29274 1/20 0.32
GSK3A P49840 1/20 0.31
GSK3B P49841 1/20 0.31
LATS1 O95835 1/20 0.31
CYP3A4 P08684 1/20 0.31
ALDH1A1 P00352 2/20 0.31
CHRNA7 P36544 2/20 0.31
CHRNB2 P17787 2/20 0.31
CHRNB4 P30926 2/20 0.31
CHRNA3 P32297 2/20 0.31
CHRNA4 P43681 2/20 0.31
CHRNA2 Q15822 2/20 0.31
MAPT P10636 2/20 0.31
LMNA P02545 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7977458 0.84 HDAC1 (0.37) GAAHDAC1CYP11B1CYP11B2ADORA3
SCHEMBL24800360 0.81 HTR2A (0.35) GAACYP11B1CYP11B2LATS1CYP3A4
SCHEMBL24669482 0.76 USP2 (0.32) GSK3BCYP3A4
SCHEMBL4013751 0.72 BRPF1 (0.50) GAAHDAC1ADORA3ALDH1A1MAPT
SCHEMBL12396551 0.71 GAA (0.40) GAACYP11B1CYP11B2ADORA3ADORA2A
SCHEMBL7975285 0.71 PDE9A (0.32) CHRNB2CHRNA4
SCHEMBL20011113 0.71 CDC7 (0.39) CYP11B1CYP11B2ADORA3ADORA2AGSK3A
SCHEMBL20571451 0.71 BRPF1 (0.62) CYP11B1CYP11B2ADORA3ADORA2AGSK3A
SCHEMBL7273301 0.69 CYP3A4 (0.32) HDAC1CYP3A4CHRNA7CHRNB2CHRNB4
SCHEMBL261618 0.68 CYP3A4 (0.40) GAACYP11B1CYP11B2CYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009147476-A1 NOVEL PDE INHIBITORS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-12-10 WO disclosed