SCHEMBL246708

SCHEMBL246708

Fc1ccc(Br)c(Br)c1F

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.39
CES1 P23141 2/20 0.39
BCHE P06276 1/20 0.32
KDM1A O60341 4/20 0.31
KCNH2 Q12809 4/20 0.31
KDM1B Q8NB78 3/20 0.31
GPR84 Q9NQS5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL313506 0.81 CES2 (0.36) CES2CES1GPR84
SCHEMBL29487566 0.81 CES2 (0.36) CES2CES1GPR84
SCHEMBL2842027 0.79 AKR1B1 (0.35) KDM1AKCNH2KDM1B
SCHEMBL29544666 0.79 KDM1A (0.41) CES2CES1KDM1AKCNH2KDM1B
SCHEMBL577838 0.79 KDM1A (0.41) CES2CES1KDM1AKCNH2KDM1B
SCHEMBL13738335 0.78 KDM1A (0.34) CES2CES1KDM1AKCNH2KDM1B
SCHEMBL1770614 0.77 KDM1A (0.35) KDM1AKCNH2KDM1B
SCHEMBL29365299 0.77 KDM1A (0.35) KDM1AKCNH2KDM1B
SCHEMBL11131552 0.72 TP53 (0.32) CES2CES1
SCHEMBL112218 0.72 HDAC4 (0.36) CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 43 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118638155-A Benzoxepin compound, preparation method and application thereof 黑龙江大学 2024-09-13 CN claimed
US-10598641-B2 Methods for determining instrument linearity and quantification THERMO FINNIGAN LLC (US) 2020-03-24 US claimed
US-20190195843-A1 METHODS FOR DETERMINING INSTRUMENT LINEARITY AND QUANTIFICATION THERMO FINNIGAN LLC 2019-06-27 US claimed
CN-118638155-A Benzoxepin compound, preparation method and application thereof 黑龙江大学 2024-09-13 CN disclosed
CN-111051284-B Compound and organic light emitting device including the same 株式会社LG化学 2023-04-18 CN disclosed
EP-3452471-B1 ORGANIC MOLECULES, ESPECIALLY FOR USE IN OPTOELECTRONIC DEVICES CYNORA GMBH (DE) 2021-12-08 EP disclosed
CN-109071501-B Organic molecules, in particular for organic opto-electronic devices 辛诺拉有限公司 2021-07-09 CN disclosed
CN-111051284-A Compound and organic light emitting device including the same 株式会社LG化学 2020-04-21 CN disclosed
WO-2019190248-A9 COMPOUND AND ORGANIC LIGHT EMITTING DIODE COMPRISING SAME 주식회사 엘지화학 2020-04-02 WO disclosed
US-10598641-B2 Methods for determining instrument linearity and quantification THERMO FINNIGAN LLC (US) 2020-03-24 US disclosed
US-10598641-B2 Methods for determining instrument linearity and quantification THERMO FINNIGAN LLC (US) 2020-03-24 US disclosed
EP-1498406-A1 Novel hydronaphthalene compounds, prepared by a rhodium catalysed ring opening reaction in the presence of phosphine ligand AstraZeneca AB (SE) 2005-01-19 EP disclosed
EP-1228024-B1 NOVEL HYDRONAPHTHALENE COMPOUNDS, PREPARED BY A RHODIUM CATALYZED RING OPENING REACTION IN THE PRESENCE OF PHOSPHINE LIGAND ASTRAZENECA AB (SE) 2004-09-01 EP disclosed
US-6784210-B2 DECYCLIZATION OF OXABENZONORBORNADIENES OR AZABICYCLIC COMPOUNDS IN THE PRESENCE OF CATALYSTS TO FORM NAPHTHALENES, SUCH AS 2-METHOXY-1,2-DIHYDRONAPHTHALEN-1-OL, USED AS ANALGESICS, ANTICARCINOGENS OR VIRICIDES; CATALYSIS ASTRAZENECA AB (SE) 2004-08-31 US disclosed
US-20030144275-A1 Decyclization of oxabenzonorbornadienes or azabicyclic compounds in the presence of catalysts to form naphthalenes, such as 2-methoxy-1,2-dihydronaphthalen-1-ol, used as analgesics, anticarcinogens or viricides; catalysis ASTRAZENECA AB (SE) 2003-07-31 US disclosed
US-6525068-B1 Such as 2-pyrrolidin-1-yl-1,2-dihydro-naphthalen-1-ol; reac-tion of oxabenzonorbornadienes with nucleophiles; pain, parkinson's disease, cancer, aids ASTRAZENECA AB (SE) 2003-02-25 US disclosed
EP-1228024-A1 NOVEL HYDRONAPHTALENE COMPOUNDS, PREPARED BY A RHODIUM CATALYZED RING OPENING REACTION IN THE PRESENCE OF PHOSPHINE LIGAND AstraZeneca AB (SE) 2002-08-07 EP disclosed
WO-2001030734-A1 NOVEL HYDRONAPHTALENE COMPOUNDS, PREPARED BY A RHODIUM CATALYZED RING OPENING REACTION IN THE PRESENCE OF PHOSPHINE LIGAND ASTRAZENECA AB (SE) 2001-05-03 WO disclosed
EP-0648724-B1 Process for the preparation of 1-Bromo-3,5-difluorobenzene HOECHST AG (DE) 1997-07-30 EP disclosed
EP-0648724-A1 Process for the preparation of 1-Bromo-3,5-difluorobenzene HOECHST AKTIENGESELLSCHAFT (DE) 1995-04-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030144275-A1 Decyclization of oxabenzonorbornadienes or azabicyclic compounds in the presence of catalysts to form naphthalenes, such as 2-methoxy-1,2-dihydronaphthalen-1-ol, used as analgesics, anticarcinogens or viricides; catalysis DDT, HPD, DHODH CES2 676/4885CES1 868/4885BCHE 650/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.