SCHEMBL24671336

SCHEMBL24671336

Cc1cc(NC(=O)c2ccc(C3=CCN(C(=N)N)CC3)cc2)ccc1N1CCN(C(=N)N)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMPRSS2 O15393 7/20 0.52
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
APOBEC3A P31941 1/20 0.46
APOBEC3G Q9HC16 1/20 0.46
CHRM1 P11229 4/20 0.46
CHRM2 P08172 1/20 0.46
CHRM4 P08173 1/20 0.46
HTR1D P28221 2/20 0.45
SLC6A4 P31645 1/20 0.45
MAPT P10636 4/20 0.41
TP53 P04637 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPY2R P49146 1/20 0.41
NAMPT P43490 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41
CYP2C19 P33261 1/20 0.41
CHRM5 P08912 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24671463 0.88 TMPRSS2 (0.49) TMPRSS2NPC1RAB9ACHRM1CHRM2
SCHEMBL29802868 0.88 CHRM1 (0.42) TMPRSS2NPC1RAB9AAPOBEC3AAPOBEC3G
SCHEMBL29802886 0.88 TMPRSS2 (0.49) TMPRSS2NPC1RAB9AAPOBEC3AAPOBEC3G
SCHEMBL29803358 0.88 TMPRSS2 (0.47) TMPRSS2NPC1RAB9AAPOBEC3AAPOBEC3G
SCHEMBL29802900 0.88 MAPT (0.43) TMPRSS2NPC1RAB9AAPOBEC3AAPOBEC3G
SCHEMBL24670017 0.88 MAPT (0.43) TMPRSS2NPC1RAB9AAPOBEC3AAPOBEC3G
SCHEMBL24671567 0.86 TP53 (0.47) TMPRSS2MAPTTP53SMN1; SMN2NPY2R
SCHEMBL29802891 0.86 APOBEC3A (0.49) TMPRSS2RAB9AAPOBEC3AAPOBEC3GCHRM1
SCHEMBL24671380 0.84 MAPT (0.53) TMPRSS2NPC1RAB9AMAPTTP53
SCHEMBL29802911 0.84 TMPRSS2 (0.41) TMPRSS2NPC1RAB9AMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO claimed
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed