SCHEMBL24671418

SCHEMBL24671418

CN1CC=C(c2ccc(C(=O)Nc3ccc(CCCNC(=N)N)cc3)s2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.39
RXFP1 Q9HBX9 1/20 0.36
ROCK2 O75116 5/20 0.36
AKT3 Q9Y243 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
USP2 O75604 2/20 0.36
ESRRG P62508 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MAPT P10636 2/20 0.35
SPHK1 Q9NYA1 4/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
ESR1 P03372 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24671416 0.90 TP53 (0.37) TP53RXFP1AKT3SMN1; SMN2USP2
Trifluoroacetic Acid SCHEMBL29803711 0.85 TP53 (0.36) TP53RXFP1AKT3SMN1; SMN2USP2
SCHEMBL24671549 0.79 TP53 (0.40) TP53RXFP1ROCK2SMN1; SMN2ESRRG
SCHEMBL24671339 0.75 MAPT (0.41) RXFP1SMN1; SMN2ESRRGNPC1MAPT
SCHEMBL29803264 0.75 RXFP1 (0.34) TP53RXFP1SMN1; SMN2ESRRGNPC1
SCHEMBL24669980 0.74 RXFP1 (0.34) TP53RXFP1SMN1; SMN2ESRRGNPC1
SCHEMBL29803084 0.72 ESRRG (0.46) RXFP1SMN1; SMN2ESRRGNPC1RAB9A
SCHEMBL24892106 0.72 ALDH1A1 (0.46) TP53SMN1; SMN2NPC1RAB9AL3MBTL1
SCHEMBL24671076 0.71 PTPN11 (0.38)
SCHEMBL24671165 0.71 ALDH1A1 (0.36) SMN1; SMN2NPC1RAB9AL3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed