SCHEMBL2467186

SCHEMBL2467186

CNc1ccnc(N(c2ccc(OC)c(S(C)(=O)=O)c2)c2n[nH]c3c(F)cccc23)n1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2D6 P10635 1/20 0.33
SCN9A Q15858 2/20 0.32
NR3C1 P04150 1/20 0.32
NR1H2 P55055 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
GAA P10253 1/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32
MAPT P10636 2/20 0.31
LMNA P02545 1/20 0.31
POLB P06746 1/20 0.31
PI4KB Q9UBF8 1/20 0.31
NR1H3 Q13133 1/20 0.30
ALOX15 P16050 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2464784 0.84 SLC40A1 (0.33) ALDH1A1CYP1A2CYP3A4SCN9AALOX15
SCHEMBL14634235 0.73 EPHB4 (0.43) CYP1A2CYP3A4CYP2D6PI4KB
SCHEMBL2466363 0.67 CHEK1 (0.36)
SCHEMBL14634005 0.67 LRRK2 (0.42)
SCHEMBL14633696 0.66 KDR (0.45) CYP1A2CYP3A4CYP2D6KMT2API4KB
SCHEMBL2469140 0.66
SCHEMBL2464853 0.65 EED (0.30)
SCHEMBL2463536 0.65 ADORA3 (0.40)
SCHEMBL14634068 0.62 EPHB4 (0.47) CYP3A4CYP2D6
SCHEMBL14633956 0.62 ABCB11 (0.53) CYP1A2CYP3A4CYP2D6PI4KB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011120025-A1 INDAZOLYL-PYRIMIDINES AS KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2011-09-29 WO disclosed