SCHEMBL24674966

SCHEMBL24674966

CCc1nc(C(F)(F)F)cnc1O

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 8/20 0.36
HCRTR2 O43614 1/20 0.34
JUN P05412 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
MTOR P42345 2/20 0.32
PIK3CA P42336 1/20 0.32
TRPV4 Q9HBA0 1/20 0.31
HEXA P06865 1/20 0.30
HEXB P07686 1/20 0.30
TRPV3 Q8NET8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25163413 0.79 HCRTR1 (0.34) HCRTR1HCRTR2JUNNFKB1NFKB2
SCHEMBL30206058 0.78 HEXA (0.40) HCRTR1HCRTR2MTORPIK3CAHEXA
SCHEMBL31336794 0.75 GAA (0.36) HCRTR1TRPV4
SCHEMBL24675335 0.71 TRPV4 (0.33) TRPV4
SCHEMBL11223672 0.71 CCR4 (0.38)
SCHEMBL22877075 0.67 HCRTR1 (0.51) HCRTR1HCRTR2
SCHEMBL30851661 0.67 USP7 (0.34) PIK3CATRPV4
SCHEMBL27223206 0.67 PDXK (0.34)
SCHEMBL16248176 0.67 JUN (0.35) JUNNFKB1NFKB2RELAHEXA
SCHEMBL24675607 0.67 TRPV4 (0.31) TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022223022-A1 FUSED-RING HETEROCYCLE DERIVATIVE AND MEDICAL APPLICATION THEREOF 四川海思科制药有限公司 2022-10-27 WO disclosed