SCHEMBL24675040

SCHEMBL24675040

CN1CCN2c3ncc(C(C)(C)C)cc3N(C)C(=O)[C@H]2C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TIPARP Q7Z3E1 4/20 0.40
HTR2A P28223 5/20 0.34
HTR2C P28335 4/20 0.34
HTR2B P41595 4/20 0.34
CYP1A2 P05177 2/20 0.34
CHRM2 P08172 2/20 0.34
HTR1A P08908 2/20 0.34
ADRA2A P08913 2/20 0.34
CYP2D6 P10635 2/20 0.34
CHRM1 P11229 2/20 0.34
CYP2C9 P11712 2/20 0.34
TSHR P16473 2/20 0.34
ADRA2B P18089 2/20 0.34
ADRA2C P18825 2/20 0.34
DRD1 P21728 2/20 0.34
CYP2C19 P33261 2/20 0.34
HTR7 P34969 2/20 0.34
ADRA1A P35348 2/20 0.34
HRH1 P35367 2/20 0.34
DRD3 P35462 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26958203 0.89 TIPARP (0.48) TIPARPHTR2AHTR2CHTR2BLMNA
SCHEMBL24675022 0.87 ALDH1A1 (0.34) TIPARPHTR2AHTR2CHTR2BCYP1A2
SCHEMBL24675034 0.87 ALDH1A1 (0.34) TIPARPHTR2AHTR2CHTR2BCYP1A2
SCHEMBL24675031 0.84 PIK3CA (0.35) TIPARPHTR2AHTR2CHTR2BCYP1A2
SCHEMBL24675038 0.83 VRK1 (0.36) TIPARPHTR2AHTR2CHTR2BCYP1A2
SCHEMBL24675049 0.81 KDM4E (0.32) TIPARPSMN1; SMN2KDM4EUSP2KMT2A
SCHEMBL24675026 0.81 TIPARP (0.33) TIPARPTSHRSMN1; SMN2KDM4EUSP2
SCHEMBL24675039 0.78 KMT2A (0.46) TIPARPHTR2AHTR2CHTR2BCYP1A2
SCHEMBL24675069 0.78 HTR2A (0.37) HTR2AHTR2CHTR2BCYP1A2CHRM2
SCHEMBL24640367 0.77 TIPARP (0.47) TIPARPCYP1A2LMNASMN1; SMN2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022223022-A1 FUSED-RING HETEROCYCLE DERIVATIVE AND MEDICAL APPLICATION THEREOF 四川海思科制药有限公司 2022-10-27 WO disclosed