SCHEMBL2467541

SCHEMBL2467541

COc1c(Cl)ccc(-c2cc(N)c(Cl)c(OC(=O)O)n2)c1F

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
HSD17B10 Q99714 1/20 0.37
MEP1B Q16820 1/20 0.34
ALOX5AP P20292 4/20 0.34
FEN1 P39748 4/20 0.34
PDCD1LG2 Q9BQ51 4/20 0.34
CD274 Q9NZQ7 4/20 0.34
HSP90AA1 P07900 2/20 0.33
HSP90AB1 P08238 2/20 0.33
FFAR4 Q5NUL3 1/20 0.32
TSHR P16473 1/20 0.32
SCN10A Q9Y5Y9 1/20 0.32
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32
TAS1R2 Q8TE23 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2468243 0.93 ALDH1A1 (0.38) ALDH1A1KDM4EHSD17B10PDCD1LG2CD274
SCHEMBL17797218 0.92 PDCD1LG2 (0.37) ALOX5APFEN1PDCD1LG2CD274HSP90AA1
SCHEMBL2468810 0.91 PDCD1LG2 (0.33) ALOX5APFEN1PDCD1LG2CD274HSP90AA1
SCHEMBL2470475 0.90 ALOX5AP (0.46) HSD17B10ALOX5APFEN1PDCD1LG2CD274
SCHEMBL2468807 0.90 MEP1B (0.36) ALDH1A1KDM4EHSD17B10MEP1BALOX5AP
SCHEMBL2465298 0.89 ALOX5AP (0.37) ALOX5APFEN1PDCD1LG2CD274FFAR4
SCHEMBL3454208 0.89 ALOX5AP (0.37) ALOX5APFEN1PDCD1LG2CD274FFAR4
SCHEMBL2463884 0.89 ALOX5AP (0.38) KDM4EALOX5APFEN1FFAR4
SCHEMBL17797261 0.88 PDCD1LG2 (0.40) PDCD1LG2CD274HSP90AA1HSP90AB1
SCHEMBL2469850 0.88 PPARA (0.33) HSP90AA1HSP90AB1FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 64 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3079473-B1 SELECTIVE WEED CONTROL WITH HALAUXIFEN DOW AGROSCIENCES LLC (US) 2020-11-11 EP claimed
EP-2947991-B1 SELECTIVE WEED CONTROL METHODS DOW AGROSCIENCES LLC (US) 2019-03-20 EP claimed
EP-2947988-B9 HERBICIDAL COMPOSITIONS COMPRISING 4-AMINO-3-CHLORO-6-(4-CHLORO-2-FLUORO-3-METHOXYPHENYL)PYRIDINE-2-CARBOXYLIC ACID DOW AGROSCIENCES LLC (US) 2019-01-23 EP claimed
EP-2947988-B1 HERBICIDAL COMPOSITIONS COMPRISING 4-AMINO-3-CHLORO-6-(4-CHLORO-2-FLUORO-3-METHOXYPHENYL)PYRIDINE-2-CARBOXYLIC ACID DOW AGROSCIENCES LLC (US) 2018-07-25 EP claimed
EP-2635116-B1 CONTROL OF PHENOXYALKANOIC ACID HERBICIDE-RESISTANT WEEDS WITH 4-AMINO-3-CHLORO-6-(4-CHLORO-2-FLUORO-3-METHOXYPHENYL)PYRIDINE-2-CARBOXYLIC ACID AND ITS SALTS OR ESTERS DOW AGROSCIENCES LLC (US) 2017-10-11 EP claimed
EP-2060566-B1 Poly-substituted aryls DOW AGROSCIENCES LLC (US) 2016-06-08 EP claimed
EP-2571366-A1 HERBICIDAL AGENTS FOR TOLERANT OR RESISTANT CORN CULTURES Bayer Intellectual Property GmbH (DE) 2013-03-27 EP claimed
EP-2571365-A1 HERBICIDAL AGENTS FOR TOLERANT OR RESISTANT GRAIN CULTURES Bayer Intellectual Property GmbH (DE) 2013-03-27 EP claimed
EP-2571363-A1 HERBICIDAL AGENTS FOR TOLERANT OR RESISTANT RAPE CULTURES Bayer Intellectual Property GmbH (DE) 2013-03-27 EP claimed
EP-2571364-A1 HERBICIDAL AGENTS FOR TOLERANT OR RESISTANT RICE CULTURES Bayer Intellectual Property GmbH (DE) 2013-03-27 EP claimed
EP-2524602-A1 Herbicide agent for tolerant or resistant soya cultures Bayer CropScience AG (DE) 2012-11-21 EP claimed
WO-2011144685-A1 HERBICIDAL AGENTS FOR TOLERANT OR RESISTANT GRAIN CULTURES BAYER CROPSCIENCE AG (DE) 2011-11-24 WO claimed
WO-2011144683-A1 HERBICIDAL AGENTS FOR TOLERANT OR RESISTANT RAPE CULTURES BAYER CROPSCIENCE AG (DE) 2011-11-24 WO claimed
WO-2011144684-A1 HERBICIDAL AGENTS FOR TOLERANT OR RESISTANT RICE CULTURES BAYER CROPSCIENCE AG (DE) 2011-11-24 WO claimed
WO-2011144691-A1 HERBICIDAL AGENTS FOR TOLERANT OR RESISTANT CORN CULTURES BAYER CROPSCIENCE AG (DE) 2011-11-24 WO claimed
WO-2010136146-A2 SYNERGISTIC COMBINATIONS OF HERBICIDES COMPRISING TEMBOTRIONE BAYER CROPSCIENCE AG (DE) 2010-12-02 WO claimed
WO-2010136165-A2 HERBICIDE COMBINATIONS COMPRISING TEFURYLTRIONE FOR USE IN RICE CULTURES BAYER CROPSCIENCE AG (DE) 2010-12-02 WO claimed
EP-2947985-B1 HERBICIDAL COMPOSITIONS COMPRISING 4-AMINO-3-CHLORO-6-(4-CHLORO-2-FLUORO-3-METHOXYPHENYL) PYRIDINE-2-CARBOXYLIC ACID DOW AGROSCIENCES LLC (US) 2019-04-03 EP disclosed
WO-2010060578-A2 HERBICIDE/SAFENER COMBINATION BAYER CROPSCIENCE AG (DE) 2010-06-03 WO disclosed
EP-2191719-A1 Herbicide safener combination Bayer CropScience AG (DE) 2010-06-02 EP disclosed