SCHEMBL24676824

SCHEMBL24676824

CC(C)c1nc(C(F)(F)F)c(-c2cc(NC3CCN(S(C)(=O)=O)CC3)ncc2F)s1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 1/20 0.43
CDK2 P24941 15/20 0.41
CCNE1 P24864 14/20 0.41
CDK1 P06493 3/20 0.41
CCNB1 P14635 2/20 0.41
CCNE2 O96020 2/20 0.41
CCNB2 O95067 1/20 0.41
CDK5 Q00535 1/20 0.41
CDK5R1 Q15078 1/20 0.41
CCNB3 Q8WWL7 1/20 0.41
GPR119 Q8TDV5 1/20 0.40
CCND1 P24385 9/20 0.39
CDK6 Q00534 9/20 0.39
RORC P51449 1/20 0.39
IDO1 P14902 1/20 0.39
CDK4 P11802 4/20 0.39
CCND3 P30281 4/20 0.39
IDH1 O75874 1/20 0.38
IDH2 P48735 1/20 0.38
CCNA2 P20248 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24677024 0.88 TDO2 (0.45) TDO2CDK2CCNE1CDK1CCNB1
SCHEMBL24676950 0.87 TDO2 (0.42) TDO2CDK2CCNE1CDK1CCNB1
SCHEMBL29754964 0.86 CDK2 (0.49) TDO2CDK2CCNE1CDK1CCNB1
SCHEMBL24676002 0.86 CDK2 (0.49) TDO2CDK2CCNE1CDK1CCNB1
SCHEMBL24676472 0.85 TDO2 (0.42) TDO2CDK2CCNE1CDK1CCNB1
SCHEMBL29754809 0.84 GPR119 (0.42) TDO2CDK2CCNE1CDK1CCNB1
SCHEMBL24676701 0.84 GPR119 (0.42) TDO2CDK2CCNE1CDK1CCNB1
SCHEMBL24676057 0.83 CDK2 (0.56) CDK2CCNE1CDK1CCNB1CCNE2
SCHEMBL24676702 0.83 GPR119 (0.40) TDO2CDK2CCNE1CDK1CCNB1
SCHEMBL24676665 0.81 GPR119 (0.40) TDO2CDK2CCNE1CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022155941-A1 CDK2 INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2022-07-28 WO disclosed