SCHEMBL24676472

SCHEMBL24676472

CS(=O)(=O)N1CCC(Nc2cc(-c3sc(CO)nc3C(F)(F)F)c(F)cn2)CC1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 1/20 0.42
GPR119 Q8TDV5 1/20 0.41
CDK2 P24941 16/20 0.40
CCNE1 P24864 14/20 0.40
CCND1 P24385 12/20 0.40
CDK6 Q00534 10/20 0.40
CDK1 P06493 6/20 0.40
CCNB1 P14635 4/20 0.40
CCNB2 O95067 1/20 0.40
CCNE2 O96020 1/20 0.40
CDK5 Q00535 1/20 0.40
CDK5R1 Q15078 1/20 0.40
CCNB3 Q8WWL7 1/20 0.40
CDK4 P11802 6/20 0.40
CCND3 P30281 4/20 0.40
CCNT1 O60563 2/20 0.39
CDK9 P50750 1/20 0.39
IDO1 P14902 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29754809 0.90 GPR119 (0.42) TDO2GPR119CDK2CCNE1CCND1
SCHEMBL24676701 0.90 GPR119 (0.42) TDO2GPR119CDK2CCNE1CCND1
SCHEMBL24676702 0.89 GPR119 (0.40) TDO2GPR119CDK2CCNE1CCND1
SCHEMBL24676665 0.87 GPR119 (0.40) TDO2GPR119CDK2CCNE1CCND1
SCHEMBL24676950 0.86 TDO2 (0.42) TDO2GPR119CDK2CCNE1CCND1
SCHEMBL24676473 0.86 RORC (0.35) CCNT1
SCHEMBL24676002 0.85 CDK2 (0.49) TDO2GPR119CDK2CCNE1CCND1
SCHEMBL24676824 0.85 TDO2 (0.43) TDO2GPR119CDK2CCNE1CCND1
SCHEMBL29754964 0.85 CDK2 (0.49) TDO2GPR119CDK2CCNE1CCND1
SCHEMBL24676489 0.83 CDK2 (0.55) CDK2CCNE1CCND1CDK6CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022155941-A1 CDK2 INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2022-07-28 WO disclosed
WO-2022155941-A1 CDK2 INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2022-07-28 WO disclosed