SCHEMBL24676665

SCHEMBL24676665

CC(C)(C)[Si](C)(C)OCc1nc(C(F)(F)F)c(-c2cc(NC3CCN(S(C)(=O)=O)CC3)ncc2F)s1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 1/20 0.40
TDO2 P48775 1/20 0.38
CDK2 P24941 15/20 0.37
CCNE1 P24864 14/20 0.37
CDK1 P06493 5/20 0.37
CCNB1 P14635 4/20 0.37
CCNB2 O95067 1/20 0.37
CCNE2 O96020 1/20 0.37
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
CCND1 P24385 10/20 0.36
CDK6 Q00534 9/20 0.36
CDK4 P11802 7/20 0.36
CCND3 P30281 4/20 0.36
CCNT1 O60563 1/20 0.35
IDO1 P14902 1/20 0.35
CCR6 P51684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24676702 0.90 GPR119 (0.40) GPR119TDO2CDK2CCNE1CDK1
SCHEMBL24676472 0.87 TDO2 (0.42) GPR119TDO2CDK2CCNE1CDK1
SCHEMBL24676701 0.85 GPR119 (0.42) GPR119TDO2CDK2CCNE1CDK1
SCHEMBL29754809 0.85 GPR119 (0.42) GPR119TDO2CDK2CCNE1CDK1
SCHEMBL24676759 0.85 CDK2 (0.51) CDK2CCNE1CDK1CCNB1CCNB2
SCHEMBL24676950 0.82 TDO2 (0.42) GPR119TDO2CDK2CCNE1CDK1
SCHEMBL24676824 0.81 TDO2 (0.43) GPR119TDO2CDK2CCNE1CDK1
SCHEMBL24676002 0.81 CDK2 (0.49) GPR119TDO2CDK2CCNE1CDK1
SCHEMBL29754964 0.81 CDK2 (0.49) GPR119TDO2CDK2CCNE1CDK1
SCHEMBL24676437 0.80 CCNE1 (0.50) CDK2CCNE1CDK1CCNB1CCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022155941-A1 CDK2 INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2022-07-28 WO disclosed