SCHEMBL24676829

SCHEMBL24676829

CNc1nc(C)c(-c2cc(NC3CCN(S(=O)(=O)C4CCNCC4)CC3)ncc2C#N)s1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 19/20 0.43
CCNA2 P20248 19/20 0.43
CDK2 P24941 19/20 0.43
CDK9 P50750 19/20 0.43
CDK1 P06493 12/20 0.43
CCNB1 P14635 12/20 0.43
CDK7 P50613 12/20 0.43
CCNH P51946 12/20 0.43
CCNA1 P78396 10/20 0.43
CCR6 P51684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24676825 0.88 CCNA2 (0.43) CCNT1CCNA2CDK2CDK9CDK1
SCHEMBL24676831 0.81 CDK9 (0.55) CCNT1CCNA2CDK2CDK9CDK1
SCHEMBL24676488 0.81 CDK2 (0.48) CCNT1CCNA2CDK2CDK9CDK1
SCHEMBL24676827 0.80 CDK2 (0.42) CCNT1CCNA2CDK2CDK9CDK1
SCHEMBL29754970 0.77 CCR6 (0.40) CCNT1CCNA2CDK2CDK9CDK1
SCHEMBL24676010 0.77 CCR6 (0.40) CCNT1CCNA2CDK2CDK9CDK1
SCHEMBL24675990 0.76 CDK2 (0.38) CCNT1CCNA2CDK2CDK9CDK1
SCHEMBL29754870 0.76 CDK2 (0.38) CCNT1CCNA2CDK2CDK9CDK1
SCHEMBL24676487 0.76 TDO2 (0.41) CCNT1CCNA2CDK2CDK9CDK1
SCHEMBL24676947 0.75 CDK2 (0.49) CCNT1CCNA2CDK2CDK9CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022155941-A1 CDK2 INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2022-07-28 WO disclosed