SCHEMBL24699353

SCHEMBL24699353

Cc1ccc(-c2nc(N3CC[C@@H]3C)nc3c2CCC3)cc1C(N)=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.39
PDK2 Q15119 1/20 0.39
PDK3 Q15120 1/20 0.39
PDK4 Q16654 1/20 0.39
GFER P55789 1/20 0.36
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP1A2 P05177 1/20 0.36
GAA P10253 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.36
GBA1 P04062 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
MTOR P42345 4/20 0.34
VCP P55072 5/20 0.34
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30015382 1.00 PDK1 (0.39) PDK1PDK2PDK3PDK4GFER
SCHEMBL30015877 0.88 PDK1 (0.40) PDK1PDK2PDK3PDK4GFER
SCHEMBL30016341 0.88 MTOR (0.44) PDK1PDK2PDK3PDK4GFER
SCHEMBL24699474 0.88 MTOR (0.44) PDK1PDK2PDK3PDK4GFER
SCHEMBL24699461 0.88 PDK1 (0.40) PDK1PDK2PDK3PDK4GFER
SCHEMBL24699484 0.86 PDE7A (0.41) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL30015689 0.86 PDE7A (0.41) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL24698594 0.86 MEN1 (0.39) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL29134886 0.86 MEN1 (0.39) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL30015817 0.86 MEN1 (0.39) PDK1PDK2PDK3PDK4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed