SCHEMBL24699461

SCHEMBL24699461

C[C@H]1CCN1c1nc2c(c(-c3ccc(C(N)=O)c(Cl)c3)n1)CCC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 2/20 0.40
PDK2 Q15119 2/20 0.40
PDK3 Q15120 2/20 0.40
PDK4 Q16654 2/20 0.40
SIRT1 Q96EB6 2/20 0.36
SIRT2 Q8IXJ6 1/20 0.36
MTOR P42345 2/20 0.36
PIK3CD O00329 1/20 0.36
ABL1 P00519 1/20 0.36
EGFR P00533 1/20 0.36
HCK P08631 1/20 0.36
SRC P12931 1/20 0.36
KDR P35968 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
EPHB4 P54760 1/20 0.36
PRKDC P78527 1/20 0.36
PI4KB Q9UBF8 1/20 0.36
MKNK1 Q9BUB5 1/20 0.35
MKNK2 Q9HBH9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30015877 1.00 PDK1 (0.40) PDK1PDK2PDK3PDK4SIRT1
SCHEMBL24699474 0.88 MTOR (0.44) PDK1PDK2PDK3PDK4SIRT1
SCHEMBL30016341 0.88 MTOR (0.44) PDK1PDK2PDK3PDK4SIRT1
SCHEMBL30015382 0.88 PDK1 (0.39) PDK1PDK2PDK3PDK4SIRT1
SCHEMBL24699353 0.88 PDK1 (0.39) PDK1PDK2PDK3PDK4SIRT1
SCHEMBL24699484 0.87 PDE7A (0.41) PDK1PDK2PDK3PDK4MTOR
SCHEMBL30015689 0.87 PDE7A (0.41) PDK1PDK2PDK3PDK4MTOR
SCHEMBL24698763 0.86 PDK1 (0.39) PDK1PDK2PDK3PDK4MTOR
SCHEMBL30016009 0.86 PDK1 (0.39) PDK1PDK2PDK3PDK4MTOR
SCHEMBL24698163 0.85 PDK2 (0.36) PDK1PDK2PDK3PDK4SIRT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed