SCHEMBL24699474

SCHEMBL24699474

C[C@H]1CCN1c1nc2c(c(-c3ccc(C(N)=O)c(F)c3)n1)CCC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 3/20 0.44
MAPK1 P28482 1/20 0.41
PDK1 Q15118 1/20 0.40
PDK2 Q15119 1/20 0.40
PDK3 Q15120 1/20 0.40
PDK4 Q16654 1/20 0.40
KDM1A O60341 1/20 0.38
PDE10A Q9Y233 2/20 0.36
PDE2A O00408 1/20 0.36
ACVR1 Q04771 2/20 0.36
GFER P55789 1/20 0.35
SIRT1 Q96EB6 1/20 0.35
PIK3CA P42336 2/20 0.34
PIK3CD O00329 1/20 0.34
HTR1A P08908 1/20 0.34
PIK3R1 P27986 1/20 0.34
PIK3CB P42338 1/20 0.34
PIK3CG P48736 1/20 0.34
DYRK1A Q13627 1/20 0.34
DYRK1B Q9Y463 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30016341 1.00 MTOR (0.44) MTORMAPK1PDK1PDK2PDK3
SCHEMBL24699461 0.88 PDK1 (0.40) MTORPDK1PDK2PDK3PDK4
SCHEMBL30015877 0.88 PDK1 (0.40) MTORPDK1PDK2PDK3PDK4
SCHEMBL24699479 0.88 ALDH1A1 (0.36) MTORPDK1PDK2PDK3PDK4
SCHEMBL30015382 0.88 PDK1 (0.39) MTORPDK1PDK2PDK3PDK4
SCHEMBL24699353 0.88 PDK1 (0.39) MTORPDK1PDK2PDK3PDK4
SCHEMBL30016009 0.88 PDK1 (0.39) MTORPDK1PDK2PDK3PDK4
SCHEMBL24698763 0.88 PDK1 (0.39) MTORPDK1PDK2PDK3PDK4
SCHEMBL24699484 0.87 PDE7A (0.41) MTORMAPK1PDK1PDK2PDK3
SCHEMBL30015689 0.87 PDE7A (0.41) MTORMAPK1PDK1PDK2PDK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed