SCHEMBL24699440

SCHEMBL24699440

Nc1ccc(-c2nc(N3CCC3)nc3c2CCC3)cn1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 14/20 0.49
PIK3R1 P27986 10/20 0.47
MTOR P42345 5/20 0.47
RICTOR Q6R327 2/20 0.47
RPTOR Q8N122 2/20 0.47
MAPKAP1 Q9BPZ7 2/20 0.47
MLST8 Q9BVC4 2/20 0.47
HRH2 P25021 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
ROCK2 O75116 1/20 0.36
CNR2 P34972 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24698993 0.85 KDM4E (0.43) PIK3CAHRH2HRH3KDM4EALDH1A1
SCHEMBL29134842 0.82 PIK3CA (0.41) PIK3CAPIK3R1MTORRICTORRPTOR
SCHEMBL24699439 0.82 PIK3CA (0.41) PIK3CAPIK3R1MTORRICTORRPTOR
SCHEMBL24698938 0.81 BACE1 (0.41) PIK3CAMTORHRH2HRH3KDM4E
SCHEMBL24698785 0.80 KDM4E (0.50) PIK3CAPIK3R1MTORRICTORRPTOR
SCHEMBL24699477 0.79 ALDH1A1 (0.47) HRH2HRH3KDM4EALDH1A1
SCHEMBL24697795 0.79 ALDH1A1 (0.40) PIK3CAHRH2HRH3KDM4EALDH1A1
SCHEMBL24698171 0.78 ALDH1A1 (0.54) KDM4EALDH1A1
SCHEMBL24698106 0.78 HRH2 (0.39) HRH2HRH3KDM4EALDH1A1
SCHEMBL24698115 0.78 HRH2 (0.41) HRH2HRH3KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed