SCHEMBL2470168

SCHEMBL2470168

Cc1ccc(CN2C(=O)c3ccccc3C2=O)c(C)c1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.57
TSHR P16473 2/20 0.55
HPGD P15428 2/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
RPS6KA2 Q15349 1/20 0.53
TGM2 P21980 1/20 0.51
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
POLB P06746 1/20 0.50
MAPT P10636 1/20 0.48
RECQL P46063 1/20 0.48
NPSR1 Q6W5P4 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
CHRM2 P08172 1/20 0.46
TNF P01375 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5473691 0.87 MAPK1 (0.54) MAPK1TSHRHPGDL3MBTL1RPS6KA2
SCHEMBL30136662 0.84 TGM2 (0.49) MAPK1TSHRHPGDRPS6KA2TGM2
SCHEMBL2478397 0.84 P2RX7 (0.52) TSHRHPGDRPS6KA2TGM2MEN1
SCHEMBL18954741 0.83 TGM2 (0.76) TSHRTGM2POLBMAPT
SCHEMBL13575895 0.83 MAPK1 (0.50) MAPK1TSHRHPGDL3MBTL1RPS6KA2
SCHEMBL10304923 0.82 PTGS1 (0.65) TSHRHPGDRPS6KA2TGM2MEN1
SCHEMBL29820186 0.82 PTGS1 (0.65) TSHRHPGDRPS6KA2TGM2MEN1
SCHEMBL3124223 0.81 CASP3 (0.56) HPGDRPS6KA2MEN1KMT2AMAPT
SCHEMBL15486283 0.81 TGM2 (0.47) MAPK1TSHRHPGDRPS6KA2TGM2
SCHEMBL19823242 0.81 RXFP1 (0.65) MAPK1TSHRHPGDRPS6KA2TGM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1787991-B2 PYRROLO[2,3-c]PYRIDINE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE TAKEDA PHARMACEUTICALS CO (JP) 2020-06-24 EP disclosed
US-20180148446-A1 PYRROLO [2,3-c] PYRIDINE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE TAKEDA PHARMACEUTICALS CO (JP) 2018-05-31 US disclosed
EP-1787991-B1 PYRROLO[2,3-c]PYRIDINE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE TAKEDA PHARMACEUTICAL (JP) 2011-10-05 EP disclosed
US-20070293532-A1 Pyrrolo [2,3-C] Pyridine Compound, Process for Producing the Same, and Use TAKEDA PHARMACEUTICAL COMPAN6Y LIMITED (JP) 2007-12-20 US disclosed
EP-1787991-A1 PYRROLOÝ2,3-c¨PYRIDINE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE Takeda Pharmaceutical Company Limited (JP) 2007-05-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180148446-A1 PYRROLO [2,3-c] PYRIDINE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE PGA5, ATP6AP1, PPA1 MAPK1 1335/4885TSHR 2787/4885HPGD 93/4885
US-20070293532-A1 Pyrrolo [2,3-C] Pyridine Compound, Process for Producing the Same, and Use PGA5, ATP6AP1, PPA1 MAPK1 1335/4885TSHR 2787/4885HPGD 93/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.