SCHEMBL2471679

SCHEMBL2471679

Cc1onc(-c2ccccc2)c1-c1cn(-c2ccccc2)c(C(=O)O)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.50
PTGS1 P23219 3/20 0.50
MAPK14 Q16539 2/20 0.49
KMT2A Q03164 3/20 0.44
MEN1 O00255 1/20 0.44
GAA P10253 1/20 0.44
MT-CO2 P00403 3/20 0.44
ALDH1A1 P00352 1/20 0.43
MAPT P10636 3/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
LMNA P02545 1/20 0.43
CA3 P07451 1/20 0.43
ADRB2 P07550 1/20 0.43
ADRB1 P08588 1/20 0.43
CYP3A4 P08684 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
CHRM1 P11229 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2474850 0.90 NPC1 (0.46) PTGS2PTGS1MAPK14KMT2AMEN1
SCHEMBL2470928 0.89 MAPK14 (0.48) PTGS2PTGS1MAPK14KMT2AGAA
SCHEMBL2472497 0.80 MAPK14 (0.49) PTGS2PTGS1MAPK14KMT2AMEN1
SCHEMBL2470836 0.80 MAPK14 (0.48) PTGS2PTGS1MAPK14KMT2AMEN1
SCHEMBL2473829 0.79 DHODH (0.45) PTGS2PTGS1MAPK14ALDH1A1MAPT
SCHEMBL4509398 0.75 ALDH1A1 (0.50) PTGS2PTGS1MAPK14KMT2AMEN1
SCHEMBL2469050 0.75 MAPT (0.46) PTGS2PTGS1MAPK14KMT2AGAA
SCHEMBL2472887 0.74 PTGS1 (0.48) PTGS2PTGS1MAPK14KMT2AMEN1
SCHEMBL2471999 0.74 PTGS2 (0.45) PTGS2PTGS1MAPK14KMT2AMEN1
SCHEMBL2472255 0.73 PTGS2 (0.52) PTGS2PTGS1MAPK14KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968973-B1 ARYL-ISOXAZOL-4-YL-IMIDAZOLE DERIVATIVES HOFFMANN LA ROCHE (CH) 2011-10-05 EP claimed