SCHEMBL2472497

SCHEMBL2472497

COC(=O)Oc1nc(-c2c(-c3ccccc3)noc2C)cn1-c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 2/20 0.49
PTGS2 P35354 6/20 0.44
PTGS1 P23219 3/20 0.44
ALDH1A1 P00352 2/20 0.44
MAPK8 P45983 1/20 0.43
MT-CO2 P00403 3/20 0.42
MAPT P10636 3/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
NR4A2 P43354 1/20 0.39
KMT2A Q03164 2/20 0.39
GAA P10253 2/20 0.39
MEN1 O00255 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HTT P42858 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
LMNA P02545 1/20 0.38
CA3 P07451 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2470928 0.83 MAPK14 (0.48) MAPK14PTGS2PTGS1ALDH1A1MAPK8
SCHEMBL2474038 0.82 MAPT (0.44) MAPK14PTGS2PTGS1MAPTTDP1
SCHEMBL2471679 0.80 PTGS2 (0.50) MAPK14PTGS2PTGS1ALDH1A1MAPK8
SCHEMBL2470836 0.74 MAPK14 (0.48) MAPK14PTGS2PTGS1ALDH1A1MAPK8
SCHEMBL2469050 0.72 MAPT (0.46) MAPK14PTGS2PTGS1ALDH1A1MT-CO2
SCHEMBL2474850 0.72 NPC1 (0.46) MAPK14PTGS2PTGS1ALDH1A1MAPK8
SCHEMBL4495802 0.71 ALDH1A1 (0.58) MAPK14PTGS2PTGS1ALDH1A1MT-CO2
SCHEMBL2470784 0.70 MAPK14 (0.42) MAPK14PTGS2PTGS1MAPK8MAPT
SCHEMBL2473829 0.70 DHODH (0.45) MAPK14PTGS2PTGS1ALDH1A1MAPT
SCHEMBL2472887 0.70 PTGS1 (0.48) MAPK14PTGS2PTGS1ALDH1A1MT-CO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968973-B1 ARYL-ISOXAZOL-4-YL-IMIDAZOLE DERIVATIVES HOFFMANN LA ROCHE (CH) 2011-10-05 EP claimed