SCHEMBL24720518

SCHEMBL24720518

Cc1cc(-c2cn[nH]c2)cc(-c2cc(C)cc(-c3ccc(N)c(Cl)c3)c2O)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.40
RPS6KA3 P51812 2/20 0.38
ESR2 Q92731 1/20 0.38
ROCK2 O75116 2/20 0.37
AKT2 P31751 5/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
AKT1 P31749 4/20 0.34
PRKACA P17612 2/20 0.34
AKT3 Q9Y243 2/20 0.34
PRKCD Q05655 2/20 0.34
RPS6KA5 O75582 1/20 0.34
RPS6KA4 O75676 1/20 0.34
LATS1 O95835 1/20 0.34
PRKACB P22694 1/20 0.34
RPS6KB1 P23443 1/20 0.34
GRK2 P25098 1/20 0.34
ROCK1 Q13464 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14896639 0.78 ALDH1A1 (0.59) RPS6KA3ESR2ROCK2AKT2ALDH1A1
SCHEMBL24720935 0.78 ESR2 (0.43) RPS6KA3ESR2ALDH1A1CYP3A4TSHR
SCHEMBL24720519 0.77 GRM2 (0.38) RPS6KA3ROCK2ERN1PRKCQPIK3CA
SCHEMBL24720649 0.74 ESR2 (0.47) ESR2ALDH1A1CYP3A4TSHRMAPK1
SCHEMBL24720587 0.74 ESR2 (0.47) ESR2ALDH1A1CYP3A4TSHRMAPK1
SCHEMBL24720257 0.73 ESR2 (0.41) RPS6KA3ESR2ALDH1A1CYP3A4TSHR
SCHEMBL24719632 0.73 ESR2 (0.43) ESR2ALDH1A1CYP3A4TSHRMAPK1
SCHEMBL24721426 0.72 TNKS2 (0.40) ESR2ALDH1A1CYP3A4TSHRMAPK1
SCHEMBL27476106 0.68 KCNH2 (0.52) LRRK2ROCK2AKT2ALDH1A1AKT1
SCHEMBL24720574 0.68 ESR2 (0.40) ESR2ALDH1A1CYP3A4TSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022261204-A1 ANTICANCER COMPOUNDS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-12-15 WO disclosed