SCHEMBL24729940

SCHEMBL24729940

Cc1cnc2c(ccn2CC2CCC2)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
GRIN1 Q05586 1/20 0.43
KCNH2 Q12809 1/20 0.43
JAK1 P23458 4/20 0.38
KDM1A O60341 2/20 0.37
GRM2 Q14416 4/20 0.36
JAK2 O60674 1/20 0.36
TYK2 P29597 1/20 0.36
CCR1 P32246 1/20 0.35
CCR5 P51681 1/20 0.35
CCR8 P51685 1/20 0.35
MAP3K5 Q99683 1/20 0.35
PDE1C Q14123 1/20 0.34
YTHDC1 Q96MU7 1/20 0.34
GRM4 Q14833 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15339573 0.94 GRIN2B (0.41) GRIN2BCYP1A2CYP2C9CYP2C19GRIN1
SCHEMBL20731030 0.83 CYP1A2 (0.38) GRIN2BCYP1A2CYP2C9CYP2C19GRIN1
SCHEMBL23938080 0.83 GRIN2B (0.43) GRIN2BCYP1A2CYP2C9CYP2C19GRIN1
SCHEMBL15712202 0.79 PKM (0.38) GRIN2BCYP1A2CYP2C9CYP2C19GRIN1
SCHEMBL31403678 0.79 KDM4C (0.40) JAK1JAK2MAP3K5
SCHEMBL21783750 0.77 MAP3K5 (0.39) GRIN2BJAK1KDM1AGRM2JAK2
SCHEMBL21704227 0.77 CCR1 (0.42) CYP1A2CCR1CCR5CCR8
SCHEMBL21783643 0.77 GRM2 (0.40) GRIN2BJAK1KDM1AGRM2JAK2
SCHEMBL7859822 0.77 HTR7 (0.42) GRIN2BJAK1KDM1AGRM2JAK2
SCHEMBL21783728 0.76 MAP3K5 (0.36) GRIN2BJAK1KDM1AGRM2JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11524966-B1 Carboxamides as ubiquitin-specific protease inhibitors VALO HEALTH, INC. (US) 2022-12-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11524966-B1 Carboxamides as ubiquitin-specific protease inhibitors USP28, USP25, USP24 GRIN2B 3388/4885CYP1A2 2136/4885CYP2C9 3180/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.