SCHEMBL2473124

SCHEMBL2473124

CCn1c(C)cc2ccnc(Cl)c21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.43
RPS6KA5 O75582 2/20 0.40
LMNA P02545 2/20 0.35
DYRK1A Q13627 3/20 0.35
DYRK3 O43781 1/20 0.34
CLK1 P49759 1/20 0.34
CLK2 P49760 1/20 0.34
CLK3 P49761 1/20 0.34
GSK3B P49841 1/20 0.34
DYRK2 Q92630 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
DYRK4 Q9NR20 1/20 0.34
DYRK1B Q9Y463 1/20 0.34
MAPT P10636 3/20 0.33
TDP1 Q9NUW8 3/20 0.33
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.33
NSD2 O96028 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2475293 0.89 KDM4E (0.44) KDM4ERPS6KA5LMNADYRK1ADYRK3
SCHEMBL2479489 0.86 KDM4E (0.44) KDM4ELMNADYRK1ADYRK2ALDH1A1
SCHEMBL2474620 0.84 HTR2A (0.32) KDM4ELMNADYRK1ADYRK3CLK1
SCHEMBL2475184 0.83 TYMS (0.46) KDM4ELMNADYRK1AMAPTALDH1A1
SCHEMBL2476573 0.82 NOTUM (0.38) LMNAALDH1A1
SCHEMBL2476713 0.82 CASR (0.38) LMNADYRK1ADYRK3CLK1CLK2
SCHEMBL2477064 0.79 GABRA5 (0.46) KDM4EALDH1A1MEN1KMT2ACYP1A2
SCHEMBL2478685 0.79 RXFP1 (0.37) KDM4ELMNADYRK1ADYRK3CLK1
SCHEMBL24896371 0.79 GPR35 (0.46)
SCHEMBL2475307 0.78 ALDH1A1 (0.51) KDM4ELMNADYRK1ADYRK3CLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1787991-B2 PYRROLO[2,3-c]PYRIDINE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE TAKEDA PHARMACEUTICALS CO (JP) 2020-06-24 EP disclosed
US-20180148446-A1 PYRROLO [2,3-c] PYRIDINE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE TAKEDA PHARMACEUTICALS CO (JP) 2018-05-31 US disclosed
EP-1787991-B1 PYRROLO[2,3-c]PYRIDINE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE TAKEDA PHARMACEUTICAL (JP) 2011-10-05 EP disclosed
US-20070293532-A1 Pyrrolo [2,3-C] Pyridine Compound, Process for Producing the Same, and Use TAKEDA PHARMACEUTICAL COMPAN6Y LIMITED (JP) 2007-12-20 US disclosed
EP-1787991-A1 PYRROLOÝ2,3-c¨PYRIDINE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE Takeda Pharmaceutical Company Limited (JP) 2007-05-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180148446-A1 PYRROLO [2,3-c] PYRIDINE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE PGA5, ATP6AP1, PPA1 KDM4E 686/4885RPS6KA5 475/4885LMNA 3382/4885
US-20070293532-A1 Pyrrolo [2,3-C] Pyridine Compound, Process for Producing the Same, and Use PGA5, ATP6AP1, PPA1 KDM4E 686/4885RPS6KA5 475/4885LMNA 3382/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.