SCHEMBL24740396

SCHEMBL24740396

CC(C)NC(=O)c1cc2c(Cl)c(Cl)ccc2[nH]1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.57
HRH4 Q9H3N8 3/20 0.52
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
RCE1 Q9Y256 1/20 0.45
ALPL P05186 2/20 0.43
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
NLRP3 Q96P20 1/20 0.40
POLB P06746 1/20 0.40
EIF4A3 P38919 1/20 0.40
THRA P10827 1/20 0.39
THRB P10828 1/20 0.39
PYGL P06737 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA2B P29275 1/20 0.39
ADORA1 P30542 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25758815 0.86 ALOX15 (0.58) ALOX15HRH4MEN1KMT2ARCE1
SCHEMBL24028985 0.85 ALOX15 (0.53) ALOX15MEN1KMT2ARCE1ALPL
SCHEMBL25758817 0.85 KMT2A (0.54) ALOX15MEN1KMT2ARCE1KDM4E
SCHEMBL24754486 0.84 HRH4 (0.56) ALOX15HRH4KMT2AFLT3
SCHEMBL24019955 0.83 ALOX15 (0.57) ALOX15HRH4MEN1KMT2ARCE1
SCHEMBL30039640 0.81 HRH4 (0.56) HRH4ALPLKDM4EALDH1A1FLT3
SCHEMBL19331400 0.81 HRH4 (0.56) HRH4ALPLKDM4EALDH1A1FLT3
SCHEMBL24450205 0.79 ALOX15 (0.52) ALOX15MEN1KMT2ARCE1ALPL
SCHEMBL17149612 0.79 MEN1 (0.48) HRH4MEN1KMT2ARCE1ADORA2A
SCHEMBL24028983 0.78 ALOX15 (0.62) ALOX15MEN1KMT2ARCE1ALPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230212152-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF Pardes Biosciences, Inc. 2023-07-06 US disclosed
US-20230212152-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF Pardes Biosciences, Inc. 2023-07-06 US disclosed
US-20230192663-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF Pardes Biosciences, Inc. 2023-06-22 US disclosed
US-11524940-B1 Inhibitors of cysteine proteases and methods of use thereof Pardes Biosciences, Inc. (US) 2022-12-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230192663-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF CTSV, CTRL, CTSL ALOX15 1562/4885HRH4 4243/4885MEN1 4363/4885
US-11524940-B1 Inhibitors of cysteine proteases and methods of use thereof CTRL, CTSV, CTSL ALOX15 1749/4885HRH4 4013/4885MEN1 4164/4885
US-20230212152-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF CTRL, CTSL, CTSV ALOX15 1455/4885HRH4 4259/4885MEN1 4306/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.