SCHEMBL2474532

SCHEMBL2474532

O=C(Nc1ccc(C(=O)N2CCN(Cc3cccc(C(O)(C(F)(F)F)C(F)(F)F)c3)CC2)cc1)NC1CCC1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
UBE2M P61081 8/20 0.53
DCUN1D1 Q96GG9 8/20 0.53
PRKAB2 O43741 3/20 0.51
PRKAG1 P54619 3/20 0.51
PRKAA2 P54646 3/20 0.51
PRKAA1 Q13131 3/20 0.51
PRKAG3 Q9UGI9 3/20 0.51
PRKAG2 Q9UGJ0 3/20 0.51
PRKAB1 Q9Y478 3/20 0.51
FAAH O00519 1/20 0.49
ACKR3 P25106 2/20 0.48
DRD4 P21917 2/20 0.48
KMT2A Q03164 2/20 0.48
DRD2 P14416 1/20 0.48
DRD3 P35462 1/20 0.48
EPHX2 P34913 1/20 0.47
SIGMAR1 Q99720 2/20 0.47
ALDH1A1 P00352 1/20 0.46
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1512304 0.89 PRKAB2 (0.60) UBE2MDCUN1D1PRKAB2PRKAG1PRKAA2
SCHEMBL1512352 0.86 PRKAB2 (0.52) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL13626743 0.85 PRKAB2 (0.56) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL1018993 0.84 DCUN1D1 (0.47) UBE2MDCUN1D1PRKAB2PRKAG1PRKAA2
SCHEMBL12954974 0.82 DRD2 (0.47) UBE2MDCUN1D1FAAHACKR3DRD4
Hydrochloric Acid SCHEMBL1074147 0.81 ACKR3 (0.46) UBE2MDCUN1D1FAAHACKR3DRD4
SCHEMBL2474230 0.80 SIGMAR1 (0.57) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL13663267 0.80 KMT2A (0.47) UBE2MDCUN1D1FAAHACKR3DRD4
SCHEMBL12954826 0.80 ACKR3 (0.45) UBE2MDCUN1D1PRKAB2PRKAG1PRKAA2
Trifluoroacetic Acid SCHEMBL1021467 0.79 SLC2A1 (0.48) UBE2MDCUN1D1PRKAB2PRKAG1PRKAA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8357679-B2 Hexafluoroisopropanol derivatives MSD OSS B.V. (NL) 2013-01-22 US disclosed
US-8357679-B2 Hexafluoroisopropanol derivatives MSD OSS B.V. (NL) 2013-01-22 US disclosed
US-8357679-B2 Hexafluoroisopropanol derivatives MSD OSS B.V. (NL) 2013-01-22 US disclosed
EP-2297118-B1 N- (1, 1, 1, 3, 3, 3-HEXAFLUORO-2-HYDROXYPROPAN-2-YL) BENZYL-N' -ARYLCARBONYLPIPERAZ INE DERIVATIVES AS LXR MODULATORS ORGANON NV (NL) 2011-10-05 EP disclosed
EP-2297118-B1 N- (1, 1, 1, 3, 3, 3-HEXAFLUORO-2-HYDROXYPROPAN-2-YL) BENZYL-N' -ARYLCARBONYLPIPERAZ INE DERIVATIVES AS LXR MODULATORS ORGANON NV (NL) 2011-10-05 EP disclosed
US-20100029621-A1 HEXAFLUOROISOPROPANOL DERIVATIVES MERCK SHARP & DOHME B.V. (NL) 2010-02-04 US disclosed
US-20100029621-A1 HEXAFLUOROISOPROPANOL DERIVATIVES MERCK SHARP & DOHME B.V. (NL) 2010-02-04 US disclosed
US-20100029621-A1 HEXAFLUOROISOPROPANOL DERIVATIVES MERCK SHARP & DOHME B.V. (NL) 2010-02-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100029621-A1 HEXAFLUOROISOPROPANOL DERIVATIVES FFAR2, FFAR3, FFAR1 UBE2M 4092/4885DCUN1D1 4694/4885PRKAB2 2245/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.