SCHEMBL24749657

SCHEMBL24749657

CCc1ccc(C2CCCOCC2)c(C)c1C

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 3/20 0.34
CEL P19835 2/20 0.34
PDE1A P54750 1/20 0.32
PDE1C Q14123 1/20 0.32
HTR2C P28335 2/20 0.31
PARP14 Q460N5 1/20 0.31
HTR6 P50406 1/20 0.30
PDCD1 Q15116 1/20 0.30
CD274 Q9NZQ7 1/20 0.30
PIK3CB P42338 1/20 0.30
PIK3CG P48736 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27672685 0.72 HTR2C (0.42) CELHTR2CHTR6
SCHEMBL22183231 0.72 CEL (0.38) CELHTR2CHTR6
SCHEMBL14231147 0.71 PIK3CB (0.31) PDE1APDE1CPIK3CBPIK3CG
SCHEMBL22156301 0.70 PDE1A (0.41) OPRL1PDE1APDE1C
SCHEMBL21163634 0.70 HTR2C (0.46) HTR2CHTR6
SCHEMBL25926930 0.69 MAPK1 (0.42) OPRL1
SCHEMBL26530978 0.68 HTR2C (0.62) OPRL1HTR2CHTR6
SCHEMBL20777893 0.68 ALDH1A1 (0.43) OPRL1HTR2CPDCD1CD274
SCHEMBL27362265 0.68 HTR6 (0.43) OPRL1HTR2CHTR6
SCHEMBL22781622 0.66 HTR2C (0.42) OPRL1HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3672952-B1 BENZIMIDAZOLE DERIVATIVES AS ADENOSINE RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 2022-12-14 EP disclosed