Etersalate

Etersalate

SCHEMBL24764

CC(=O)Nc1ccc(OCCOC(=O)c2ccccc2OC(C)=O)cc1

nearest known ligand 0.71

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.51
LMNA P02545 4/20 0.50
PTGS2 P35354 3/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
HPGD P15428 3/20 0.50
HSD17B10 Q99714 3/20 0.50
KDM4E B2RXH2 2/20 0.49
MAPT P10636 1/20 0.49
GLA P06280 1/20 0.49
KMT2A Q03164 5/20 0.48
MEN1 O00255 3/20 0.48
TDP1 Q9NUW8 2/20 0.48
CYP1A2 P05177 1/20 0.48
NPC1 O15118 2/20 0.47
EGFR P00533 1/20 0.47
TP53 P04637 1/20 0.46
NFKB1 P19838 1/20 0.46
RAB9A P51151 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benorilate SCHEMBL15526470 0.83 HSD17B10 (0.70) ALDH1A1LMNAPTGS2SMN1; SMN2HPGD
Benorilate SCHEMBL25167 0.83 HSD17B10 (0.70) ALDH1A1LMNAPTGS2SMN1; SMN2HPGD
Benorilate SCHEMBL27446831 0.83 HSD17B10 (0.70) ALDH1A1LMNAPTGS2SMN1; SMN2HPGD
Benorilate SCHEMBL15969775 0.82 HSD17B10 (0.68) ALDH1A1LMNAPTGS2SMN1; SMN2HPGD
SCHEMBL11985691 0.82 PTGS2 (0.68) ALDH1A1LMNAPTGS2HPGDHSD17B10
SCHEMBL15079378 0.81 ALDH1A1 (0.55) ALDH1A1LMNASMN1; SMN2MAPTKMT2A
Etersalate SCHEMBL19025606 0.80 KMT2A (0.48) ALDH1A1LMNAHPGDHSD17B10KDM4E
Aspirin SCHEMBL10380307 0.80 KMT2A (0.63) ALDH1A1LMNAPTGS2SMN1; SMN2HPGD
Benorilate SCHEMBL1162333 0.79 HSD17B10 (0.68) ALDH1A1LMNAPTGS2SMN1; SMN2HPGD
SCHEMBL11985703 0.78 PTGS2 (0.63) ALDH1A1LMNAPTGS2SMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2444 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12194158-B2 Oromucosal nanofiber carriers for therapeutic treatment INSTAR TECHNOLOGIES A.S. (CZ) 2025-01-14 US claimed
US-20240041935-A1 PREVENTION AND TREATMENT OF REPRODUCTIVE FAILURE BY REGENERATIVE CELLS AND ADJUVANTS CREATIVE MEDICAL TECHNOLOGIES, INC. (US) 2024-02-08 US claimed
WO-2023138079-A1 PREPARATION METHOD FOR 2'-SUBSTITUTED PYRIMIDINE NUCLEOSIDE 北京瑞博奥医药科技有限公司 2023-07-27 WO claimed
US-9161927-B2 Drug combinations containing PDE4 inhibitors and NSAIDs BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-10-20 US claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-8759326-B2 Drug combinations containing PDE4 inhibitors and NSAIDs BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-06-24 US claimed
US-20140031343-A1 DRUG COMBINATIONS CONTAINING PDE4 INHIBITORS AND NSAIDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-01-30 US claimed
US-8592400-B2 Drug combinations containing PDE4 inhibitors and NSAIDs BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-11-26 US claimed
EP-2560634-A1 NITRIC OXIDE RELEASING PRODRUGS OF THERAPEUTIC AGENTS Piramal Enterprises Limited (IN) 2013-02-27 EP claimed
US-8361492-B2 Drug delivery system and methods of use Ocugenics, LLC (US) 2013-01-29 US claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
EP-0786999-A4 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO INC (US) 1999-01-20 EP claimed
EP-0792371-A4 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO INC (US) 1998-12-30 EP claimed
WO-1998020864-A9 USE OF SELECTED NON-STEROIDAL ANTIINFLAMMATORY COMPOUNDS FOR THE PREVENTION AND THE TREATMENT OF NEURODEGENERATIVE DISEASES 1998-08-27 WO claimed
WO-1998020864-A2 USE OF SELECTED NON-STEROIDAL ANTIINFLAMMATORY COMPOUNDS FOR THE PREVENTION AND THE TREATMENT OF NEURODEGENERATIVE DISEASES UNIVERSITA' DEGLI STUDI DI BRESCIA - DIPARTIMENTO DI SCIENZE BIOMEDICHE (IT) 1998-05-22 WO claimed
EP-0792371-A1 COMBINATION METHOD FOR ACNE TREATMENT Merck & Co., Inc. (US) 1997-09-03 EP claimed
EP-0786999-A1 COMBINATION METHOD FOR ACNE TREATMENT Merck & Co., Inc. (US) 1997-08-06 EP claimed
US-5543417-A 5 Alpha-reductase inhibitor and at least one of an antibacterial agent, a keratolytic agent or an anti-inflammatory agent MERCK & CO., INC. (US) 1996-08-06 US claimed
WO-1996012487-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO claimed
WO-1996012817-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO claimed