SCHEMBL24784367

SCHEMBL24784367

Cc1ccc(Nc2cc(C)nc(N3CCN(C(=O)CCc4ccccc4)CC3)n2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.54
MAPT P10636 2/20 0.54
GBA1 P04062 1/20 0.53
KDM4E B2RXH2 3/20 0.52
ALDH1A1 P00352 3/20 0.52
HPGD P15428 2/20 0.52
HSD17B10 Q99714 2/20 0.52
TSHR P16473 1/20 0.52
JAK2 O60674 1/20 0.50
CCNE1 P24864 3/20 0.49
CDK2 P24941 3/20 0.49
ALOX15 P16050 1/20 0.48
USP2 O75604 1/20 0.47
HTT P42858 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
SLC2A1 P11166 1/20 0.46
ME2 P23368 1/20 0.46
ME1 P48163 1/20 0.46
ME3 Q16798 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8354085 0.85 ALDH1A1 (0.64) MAPTGBA1KDM4EALDH1A1HPGD
SCHEMBL18153314 0.83 LMNA (0.66) LMNAMAPTGBA1KDM4EALDH1A1
SCHEMBL18063521 0.76 MAPT (0.58) LMNAMAPTKDM4EALDH1A1HPGD
SCHEMBL18087196 0.74 LMNA (0.60) LMNAMAPTGBA1KDM4EALDH1A1
SCHEMBL21015066 0.74 LMNA (0.62) LMNAMAPTGBA1KDM4EALDH1A1
SCHEMBL7176075 0.73 SMN1; SMN2 (0.71) LMNAKDM4EALDH1A1TSHRL3MBTL1
SCHEMBL18153366 0.73 MAPT (0.51) LMNAMAPTKDM4EALDH1A1HPGD
SCHEMBL3796501 0.72 MAPT (0.70) LMNAMAPTALDH1A1HSD17B10NPSR1
SCHEMBL11506640 0.72 GALR2 (0.66) LMNAMAPTKDM4ENPSR1
SCHEMBL18063516 0.71 LMNA (0.72) LMNAMAPTKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022261296-A1 COMPOUNDS THAT BIND NON-CANONICAL G-QUADRUPLEX STRUCTURES AND METHODS OF MAKING AND USING THE SAME THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2022-12-15 WO disclosed