SCHEMBL24802486

SCHEMBL24802486

CCOC(=O)Cc1nc2ccc(Br)cc2c(=O)[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.53
ALDH1A1 P00352 2/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
JAK2 O60674 1/20 0.51
PAK4 O96013 1/20 0.51
NTRK1 P04629 1/20 0.51
LCK P06239 1/20 0.51
FYN P06241 1/20 0.51
CSF1R P07333 1/20 0.51
RET P07949 1/20 0.51
MET P08581 1/20 0.51
PDGFRB P09619 1/20 0.51
PIM1 P11309 1/20 0.51
FGFR1 P11362 1/20 0.51
PRKACA P17612 1/20 0.51
GRK5 P34947 1/20 0.51
MAP2K2 P36507 1/20 0.51
FLT3 P36888 1/20 0.51
MAPK8 P45983 1/20 0.51
CDK8 P49336 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10084487 0.88 HSD17B10 (0.55) HSD17B10ALDH1A1SMN1; SMN2GAAMAPT
SCHEMBL4743261 0.82 HSD17B10 (0.69) HSD17B10ALDH1A1SMN1; SMN2GAAMAPT
SCHEMBL11548717 0.81 HSD17B10 (0.61) HSD17B10ALDH1A1SMN1; SMN2GAAMAPT
SCHEMBL12940747 0.81 HSD17B10 (0.67) HSD17B10ALDH1A1SMN1; SMN2JAK2PAK4
SCHEMBL17298090 0.80 TNKS2 (0.62) ALDH1A1SMN1; SMN2PIM1FLT3GAA
SCHEMBL8197895 0.80 ALDH1A1 (0.62) HSD17B10ALDH1A1SMN1; SMN2GAAMAPT
SCHEMBL30208243 0.80 ALDH1A1 (0.62) HSD17B10ALDH1A1SMN1; SMN2GAAMAPT
SCHEMBL3110721 0.74 KDM4E (0.56) SMN1; SMN2PIM1FLT3GAAMAPT
SCHEMBL19104692 0.74 TUBB4A (0.48) HSD17B10ALDH1A1SMN1; SMN2PIM1FLT3
SCHEMBL3840420 0.73 HSD17B10 (0.71) HSD17B10ALDH1A1SMN1; SMN2GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117580836-A Pyrimidine ring structure derivative and application thereof 四川汇宇制药股份有限公司 2024-02-20 CN disclosed
WO-2022268209-A1 DERIVATIVE HAVING PYRIMIDINE-FUSED CYCLIC STRUCTURE, AND USE THEREOF 四川汇宇制药股份有限公司 2022-12-29 WO disclosed
WO-2022268209-A1 DERIVATIVE HAVING PYRIMIDINE-FUSED CYCLIC STRUCTURE, AND USE THEREOF 四川汇宇制药股份有限公司 2022-12-29 WO disclosed