SCHEMBL2480595

SCHEMBL2480595

CC(C(=O)O)N1C(=O)C(=O)c2cc(Cl)ccc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH3A1 P30838 6/20 0.47
ALDH1A1 P00352 3/20 0.47
ALDH2 P05091 3/20 0.47
KDM4E B2RXH2 2/20 0.46
GAA P10253 1/20 0.46
CASP1 P29466 1/20 0.46
CASP7 P55210 1/20 0.46
KMT2A Q03164 1/20 0.46
AGTR1 P30556 1/20 0.40
MYC P01106 1/20 0.40
NR4A1 P22736 1/20 0.40
PDE5A O76074 1/20 0.38
ACHE P22303 1/20 0.38
HSD17B10 Q99714 1/20 0.37
CSNK2A2 P19784 1/20 0.37
CSNK2B P67870 1/20 0.37
CSNK2A1 P68400 1/20 0.37
S100A4 P26447 1/20 0.37
SDCBP O00560 1/20 0.37
SDC2 P34741 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9105740 0.83 ALDH1A1 (0.46) ALDH3A1ALDH1A1ALDH2
SCHEMBL281661 0.83 ALDH3A1 (0.48) ALDH3A1ALDH1A1ALDH2KDM4EAGTR1
SCHEMBL11192451 0.83 ALDH3A1 (0.49) ALDH3A1ALDH1A1ALDH2AGTR1S100A4
SCHEMBL2833377 0.82 CASP3 (0.54) ALDH1A1KDM4EGAACASP1CASP7
SCHEMBL18954664 0.82 KDM4E (0.46) ALDH1A1KDM4EGAACASP1CASP7
SCHEMBL2482727 0.82 ALDH3A1 (0.44) ALDH3A1ALDH1A1ALDH2AGTR1MYC
SCHEMBL18954629 0.80 KDM4E (0.44) ALDH1A1KDM4EGAACASP1CASP7
SCHEMBL18954671 0.79 KDM4E (0.43) ALDH1A1KDM4EGAACASP1CASP7
SCHEMBL18954672 0.79 KDM4E (0.43) ALDH1A1KDM4EGAACASP1CASP7
SCHEMBL18955246 0.79 CA1 (0.49) KDM4EGAACASP1CASP7KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891075-B1 TRICYCLIC SPIRO DERIVATIVES AS CRTH2 MODULATORS MERCK SERONO SA (CH) 2011-10-19 EP disclosed