SCHEMBL2482274

SCHEMBL2482274

Nc1ccc2c(c1)NC(CC=O)CCC2

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 1/20 0.45
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
BRD4 O60885 1/20 0.35
ATAD2 Q6PL18 1/20 0.35
GRIN2B Q13224 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4015772 0.91 CA9 (0.47) CA9ITGB3ITGA2BKDM4EMEN1
SCHEMBL7399575 0.82 ITGB3 (0.57) CA9ITGB3ITGA2BKDM4EMEN1
SCHEMBL7399576 0.82 ITGB3 (0.57) CA9ITGB3ITGA2BKDM4EMEN1
Methane SCHEMBL28580610 0.77 CA9 (0.44) CA9ITGB3ITGA2BKDM4EMEN1
SCHEMBL2484227 0.75 CMA1 (0.39)
SCHEMBL4967797 0.72 CA9 (0.34) CA9KDM4EMEN1GAAMAPT
SCHEMBL15263464 0.72 CA9 (0.41) CA9ITGB3ITGA2BKDM4EMEN1
SCHEMBL27771607 0.71 CA9 (0.47) CA9KDM4EMEN1GAAMAPT
SCHEMBL4017459 0.69 PNMT (0.42) GRIN2B
SCHEMBL12450086 0.68 PNMT (0.35) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376491-A1 PYRROLOTRIAZINES AS ALK AND JAK2 INHIBITORS Cephalon, Inc. (US) 2011-10-19 EP disclosed
WO-2010071885-A1 PYRROLOTRIAZINES AS ALK AND JAK2 INHIBITORS CEPHALON, INC. (US) 2010-06-24 WO disclosed