SCHEMBL24823955

SCHEMBL24823955

CC1CCc2cc(Br)cnc2NC1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.42
CRBN Q96SW2 5/20 0.35
DDB1 Q16531 2/20 0.35
PLK4 O00444 1/20 0.33
SMYD3 Q9H7B4 2/20 0.32
NNMT P40261 2/20 0.32
MB P02144 1/20 0.32
BRD4 O60885 1/20 0.32
AURKA O14965 2/20 0.32
DAPK3 O43293 2/20 0.32
PRKD3 O94806 2/20 0.32
MAP4K4 O95819 2/20 0.32
ABL1 P00519 2/20 0.32
NTRK1 P04629 2/20 0.32
RET P07949 2/20 0.32
MET P08581 2/20 0.32
PDGFRB P09619 2/20 0.32
PIM1 P11309 2/20 0.32
FGFR1 P11362 2/20 0.32
PDGFRA P16234 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2276398 0.86 AKR1B1 (0.40) AKR1B1CRBNDDB1PLK4SMYD3
SCHEMBL24723078 0.84 SMYD3 (0.36) AKR1B1CRBNDDB1PLK4SMYD3
SCHEMBL23532191 0.84 CRBN (0.35) AKR1B1CRBNDDB1PLK4SMYD3
SCHEMBL24823109 0.83 CRBN (0.37) AKR1B1CRBNDDB1PLK4SMYD3
SCHEMBL30304182 0.83 AKR1B1 (0.34) AKR1B1CRBNDDB1PLK4SMYD3
SCHEMBL24823074 0.83 AKR1B1 (0.34) AKR1B1CRBNDDB1PLK4SMYD3
SCHEMBL30304181 0.83 CRBN (0.37) AKR1B1CRBNDDB1PLK4SMYD3
SCHEMBL30160396 0.78 L3MBTL4 (0.36) CRBNDDB1HSD17B10
SCHEMBL23532125 0.78 L3MBTL4 (0.36) CRBNDDB1HSD17B10
SCHEMBL29189520 0.78 CRBN (0.33) AKR1B1CRBNDDB1SMYD3NNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230159519-A1 NOVEL COMPOUNDS AND THEIR USE DEBIOPHARM INTERNATIONAL S.A. (CH) 2023-05-25 US disclosed
US-20230159519-A1 NOVEL COMPOUNDS AND THEIR USE DEBIOPHARM INTERNATIONAL S.A. (CH) 2023-05-25 US disclosed
WO-2022268890-A1 NOVEL COMPOUNDS AND THEIR USE DEBIOPHARM INTERNATIONAL S.A. (CH) 2022-12-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230159519-A1 NOVEL COMPOUNDS AND THEIR USE LSS, PGLS, LDHB AKR1B1 1042/4885CRBN 2073/4885DDB1 1225/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.