SCHEMBL24848629

SCHEMBL24848629

CC(C)c1cc(C(F)(F)F)nc(C(C)(C)C)n1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.59
CYP2D6 P10635 1/20 0.59
TSHR P16473 1/20 0.59
CRHBP P24387 1/20 0.59
CYP2C19 P33261 1/20 0.59
CRHR2 Q13324 1/20 0.59
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
DRD2 P14416 14/20 0.33
DRD3 P35462 14/20 0.33
HMGCR P04035 2/20 0.33
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25065713 0.89 CYP2C19 (0.62) CYP3A4CYP2D6TSHRCRHBPCYP2C19
SCHEMBL16259689 0.86 HMGCR (0.42) CYP3A4CYP2D6TSHRCRHBPCYP2C19
SCHEMBL26022486 0.78 HSP90AA1 (0.41) CYP3A4CYP2D6TSHRCRHBPCYP2C19
SCHEMBL798992 0.77 CYP2C19 (0.62) CYP3A4CYP2D6TSHRCRHBPCYP2C19
SCHEMBL18068094 0.76 CYP3A4 (0.50) CYP3A4CYP2D6TSHRCRHBPCYP2C19
SCHEMBL22767093 0.76 CYP2C19 (0.61) CYP3A4CYP2D6TSHRCRHBPCYP2C19
SCHEMBL22249889 0.75 NOS3 (0.39) CYP3A4CYP2D6TSHRCRHBPCYP2C19
SCHEMBL13201505 0.75 HSP90AA1 (0.57) CYP3A4CYP2D6TSHRCRHBPCYP2C19
SCHEMBL20211619 0.74 CYP2C19 (1.00) CYP3A4CYP2D6TSHRCRHBPCYP2C19
SCHEMBL21731005 0.73 CYP2C19 (0.58) CYP3A4CYP2D6TSHRCRHBPCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230002364-A1 BENZOTHIOPHENE DERIVATIVE REGULATOR, PREPARATION METHOD THEREFOR AND USE THEREOF JIANGSU HANSOH PHARMACEUTICAL GROUP CO., LTD. (CN) 2023-01-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230002364-A1 BENZOTHIOPHENE DERIVATIVE REGULATOR, PREPARATION METHOD THEREFOR AND USE THEREOF GPER1, GABRQ, GPR39 CYP3A4 1019/4885CYP2D6 1428/4885TSHR 587/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.